SCHEMBL5323972

SCHEMBL5323972

NC(=O)c1ccc(Cl)c(C(=O)N2CCC(Cc3ccc(F)cc3)CC2)c1

nearest known ligand 0.58

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
MAPK14 Q16539 5/20 0.55
CYP2C9 P11712 2/20 0.55
CYP2C19 P33261 2/20 0.55
HTR2B P41595 1/20 0.55
HSD11B1 P28845 3/20 0.50
CCR3 P51677 1/20 0.50
PRSS12 P56730 2/20 0.49
GAA P10253 1/20 0.48
CHRM2 P08172 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5323974 0.87 MAPK14 (0.57) MAPK14CYP2C9CYP2C19HTR2BCCR3
Hydrochloric Acid SCHEMBL5321355 0.86 MAPK14 (0.56) MAPK14CYP2C9CYP2C19HTR2BCCR3
SCHEMBL5319166 0.84 MAPK14 (0.57) MAPK14CYP2C9CYP2C19HTR2BHSD11B1
SCHEMBL5323527 0.84 MAPK14 (0.76) MAPK14CYP2C9CYP2C19HSD11B1
SCHEMBL5323872 0.79 MAPK14 (0.54) MAPK14CYP2C9CYP2C19HTR2B
SCHEMBL14467025 0.76 MAPK14 (0.60) MAPK14CYP2C9CYP2C19HTR2BCCR3
SCHEMBL5346573 0.76 AURKA (0.49) MAPK14CYP2C9CYP2C19HTR2BCCR3
SCHEMBL13936069 0.76 MAPK14 (0.62) MAPK14CYP2C9CYP2C19HTR2BCCR3
SCHEMBL5806708 0.76 MEN1 (0.55) MAPK14CYP2C9CYP2C19CCR3
SCHEMBL4243148 0.75 GAA (0.55) GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007082079-A2 PIPERIDINE AMIDE DERIVATIVES AS PROTEIN KINASE INHIBITORS THE SCRIPPS RESEARCH INSTITUTE (US) 2007-07-19 WO disclosed