SCHEMBL5325844

SCHEMBL5325844

Cc1ccc2c(c1)N(c1ccc(N)cc1)C(=O)N(C1COc3ccccc3OC1)N=C2C1CCOCC1

nearest known ligand 0.58

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
PTH1R Q03431 18/20 0.58
NPC1 O15118 1/20 0.32
ALDH1A1 P00352 1/20 0.32
TSHR P16473 1/20 0.32
CASP1 P29466 1/20 0.32
RAB9A P51151 1/20 0.32
CASP7 P55210 1/20 0.32
HSD17B10 Q99714 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5323234 0.92 PTH1R (0.67) PTH1R
SCHEMBL5330610 0.87 PTH1R (0.67) PTH1R
SCHEMBL5320230 0.85 PTH1R (0.65) PTH1R
SCHEMBL5329276 0.84 PTH1R (0.51) PTH1RNPC1ALDH1A1TSHRCASP1
SCHEMBL5320434 0.84 PTH1R (0.51) PTH1RNPC1ALDH1A1TSHRCASP1
SCHEMBL5321102 0.80 PTH1R (0.57) PTH1R
SCHEMBL5323133 0.80 PTH1R (0.57) PTH1R
SCHEMBL5326711 0.80 PTH1R (0.57) PTH1R
SCHEMBL5325857 0.78 PTH1R (0.66) PTH1R
SCHEMBL5326666 0.78 PTH1R (0.54) PTH1R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006129120-A9 BENZOTRIAZEPINONE DERIVATIVES JAMES BLACK FOUNDATION (GB) 2007-03-22 WO disclosed
WO-2006129120-A2 BENZOTRIAZEPINONE DERIVATIVES JAMES BLACK FOUNDATION (GB) 2006-12-07 WO disclosed