SCHEMBL5325975

SCHEMBL5325975

Cc1ccc2c(c1)N(c1ccc(N)cc1)C(=O)N(C)N=C2C1CCCCC1

nearest known ligand 0.64

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
PTH1R Q03431 19/20 0.64
NPC1 O15118 1/20 0.39
ALDH1A1 P00352 1/20 0.39
TSHR P16473 1/20 0.39
CASP1 P29466 1/20 0.39
RAB9A P51151 1/20 0.39
CASP7 P55210 1/20 0.39
HSD17B10 Q99714 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5321102 0.88 PTH1R (0.57) PTH1R
SCHEMBL5326711 0.88 PTH1R (0.57) PTH1R
SCHEMBL5323133 0.88 PTH1R (0.57) PTH1R
SCHEMBL5319846 0.87 PTH1R (0.65) PTH1R
SCHEMBL5322629 0.87 PTH1R (0.63) PTH1R
SCHEMBL5322500 0.86 PTH1R (0.51) PTH1R
SCHEMBL5325766 0.85 PTH1R (0.59) PTH1R
SCHEMBL5282657 0.85 PTH1R (0.67) PTH1R
SCHEMBL5326346 0.84 PTH1R (0.54) PTH1R
SCHEMBL5321308 0.84 PTH1R (0.54) PTH1R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006129120-A9 BENZOTRIAZEPINONE DERIVATIVES JAMES BLACK FOUNDATION (GB) 2007-03-22 WO disclosed
WO-2006129120-A2 BENZOTRIAZEPINONE DERIVATIVES JAMES BLACK FOUNDATION (GB) 2006-12-07 WO disclosed