SCHEMBL53264

SCHEMBL53264

Cc1n[c]sc1C

nearest known ligand 0.00

⚠ Novel chemotype — no close known analogue (best Tanimoto < 0.3). Unexplored chemical space relative to ChEMBL.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3430838 0.71
SCHEMBL16341358 0.71
SCHEMBL21645374 0.71
SCHEMBL2579554 0.71
SCHEMBL8122170 0.67
SCHEMBL3186717 0.67
SCHEMBL2441506 0.66
SCHEMBL2441980 0.66
SCHEMBL9151789 0.66
SCHEMBL2440626 0.66

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1379 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024140294-A1 ORGANIC COMPOUND AND APPLICATION THEREOF IN OLED DEVICE 北京云基科技股份有限公司 2024-07-04 WO claimed
US-11950507-B2 Organic electroluminescence device Beijing Summer Sprout Technology Co., Ltd. (CN) 2024-04-02 US claimed
CN-114335361-B Composition and organic electroluminescent device comprising same 江苏三月科技股份有限公司 2024-03-22 CN claimed
CN-114335364-B Composition for organic electroluminescent device and organic electroluminescent device 江苏三月科技股份有限公司 2024-03-22 CN claimed
CN-117693217-A Series organic electroluminescent device 北京夏禾科技有限公司 2024-03-12 CN claimed
US-11897896-B2 Organic electroluminescent materials and devices Beijing Summer Sprout Technology Co., Ltd. 2024-02-13 US claimed
CN-114335362-B OLED (organic light emitting diode) composition and organic electroluminescent device 江苏三月科技股份有限公司 2024-02-13 CN claimed
CN-114335363-B Composition for organic electroluminescent device and organic electroluminescent device 江苏三月科技股份有限公司 2024-01-30 CN claimed
US-20230390259-A1 PHARMACEUTICAL COMPOSITION COMPRISING PYRIDONE DERIVATIVES SK BIOPHARMACEUTICALS CO., LTD. (KR) 2023-12-07 US claimed
US-20230348516-A1 YKL-40 INHIBITORS AND THEIR THERAPEUTIC APPLICATIONS MOLECURE S.A. (PL) 2023-11-02 US claimed
US-4187303-A ANTIINFLAMMATORY AGENTS, ANALGESICS, ANTICOAGULANTS HOFFMANN-LA ROCHE INC. (US) 1980-02-05 US claimed
US-4183856-A FROM HETEROAROMATIC SECONDARY AMINES AND CARBAMOYL HALOGENIDES IN THE PRESENCE OF A LEWIS ACID SHIONOGI & CO., LTD. (JP) 1980-01-15 US claimed
US-4180662-A ANTIINFLAMMATORY, ANALGESIC, ANTIRHEUMATIC, ANTITHROMBOTIC HOFFMANN-LA ROCHE INC. (US) 1979-12-25 US claimed
EP-0001113-A1 Thienothiazine derivatives, their preparation and compositions containing them F. HOFFMANN-LA ROCHE & CO. Aktiengesellschaft (CH) 1979-03-21 EP claimed
US-RE29669-E CYCLIZATION OF GLYCINEAMIDES PFIZER, INC. (US) 1978-06-13 US claimed
US-RE29668-E 4-OXO-1,2-BENZOTHIAZINE-3-CARBOXAMIDE, 1,1-DIOXIDES, ANTIINFLAMMATORY PFIZER INC. (US) 1978-06-13 US claimed
US-4090020-A ANTIINFLAMMATORY AGENTS, ANALGESICS, ANTIRHEUMATIC AGENTS HOFFMANN-LA ROCHE INC. (US) 1978-05-16 US claimed
US-4076709-A ANTIINFLAMMATORY AGENTS, ANALGESICS, ANTIRHEUMATIC AGENTS HOFFMANN-LA ROCHE INC. (US) 1978-02-28 US claimed
US-3992535-A ANTIINFLAMMATORY AGENTS, INHIBITORS OF PLATELET ADHESION AND AGGREGATION BOEHRINGER INGELHEIM GMBH (DT) 1976-11-16 US claimed
US-3971802-A ANTIINFLAMMATORY PFIZER INC. (US) 1976-07-27 US claimed