SCHEMBL532858

SCHEMBL532858

Cc1cc(C)c(N2CCCC2)c(C)c1NC(=O)c1sccc1S(=O)(=O)Nc1ccccc1.Cc1cc(C)c(N2CCCC2)c(C)c1NS(=O)(=O)c1ccc(Cl)cc1

nearest known ligand 0.47

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
EDNRA P25101 12/20 0.47
MEN1 O00255 3/20 0.44
KMT2A Q03164 3/20 0.44
CYP3A4 P08684 2/20 0.44
TSHR P16473 1/20 0.44
GPR27 Q9NS67 1/20 0.43
MAPT P10636 2/20 0.42
EDNRB P24530 1/20 0.42
IDH1 O75874 3/20 0.42
KDM4E B2RXH2 1/20 0.41
ALDH1A1 P00352 1/20 0.41
GAA P10253 1/20 0.41
DUSP3 P51452 1/20 0.41
PTPN5 P54829 1/20 0.41
PTPN11 Q06124 1/20 0.41
HSD17B10 Q99714 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL532974 0.92 EDNRA (0.49) EDNRAMEN1KMT2ACYP3A4MAPT
SCHEMBL3976730 0.85 EDNRA (0.42) EDNRAMEN1KMT2ACYP3A4TSHR
SCHEMBL3972434 0.83 MAPT (0.49) EDNRAMEN1KMT2AMAPTEDNRB
SCHEMBL3975239 0.83 EDNRA (0.46) EDNRAMEN1KMT2ACYP3A4MAPT
SCHEMBL532871 0.82 MEN1 (0.45) EDNRAMEN1KMT2ACYP3A4TSHR
SCHEMBL3976237 0.81 MEN1 (0.44) EDNRAMEN1KMT2ACYP3A4TSHR
SCHEMBL3977551 0.80 MEN1 (0.48) EDNRAMEN1KMT2ACYP3A4MAPT
SCHEMBL3974388 0.79 MAPT (0.49) EDNRAMEN1KMT2AMAPTEDNRB
SCHEMBL533012 0.79 MEN1 (0.56) EDNRAMEN1KMT2ACYP3A4TSHR
SCHEMBL3978595 0.79 MEN1 (0.46) EDNRAMEN1KMT2ACYP3A4MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2415760-A2 CCR-9 antagonists ENCYSIVE PHARMACEUTICALS, INC. (US) 2012-02-08 EP disclosed