SCHEMBL5329148

SCHEMBL5329148

COc1cccc(C2=NNCCC2)c1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NISCH Q9Y2I1 1/20 0.49
GAA P10253 3/20 0.48
DYRK1A Q13627 1/20 0.45
CLK4 Q9HAZ1 1/20 0.45
MAOB P27338 1/20 0.43
WDR5 P61964 1/20 0.43
MAPT P10636 3/20 0.42
RAB9A P51151 3/20 0.42
SMN1; SMN2 Q16637 3/20 0.42
ALDH1A1 P00352 2/20 0.42
KDM4E B2RXH2 2/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
KMT2A Q03164 1/20 0.42
CASP3 P42574 1/20 0.41
SENP8 Q96LD8 1/20 0.41
SENP7 Q9BQF6 1/20 0.41
SENP6 Q9GZR1 1/20 0.41
NOTUM Q6P988 1/20 0.40
NR1H2 P55055 1/20 0.40
NR1H3 Q13133 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12922944 0.91 NISCH (0.51) NISCHGAADYRK1ACLK4MAOB
SCHEMBL31309661 0.80 CHRNB4 (0.57) NISCHMAOBMAPTRAB9ASMN1; SMN2
SCHEMBL5203405 0.77 PDE4B (0.63) MAOBMAPTALDH1A1KDM4E
SCHEMBL2806024 0.76 CHRNB4 (0.57) NISCHGAADYRK1ACLK4MAOB
SCHEMBL5309374 0.75 PDE3B (0.63) GAAMAPTRAB9ASMN1; SMN2ALDH1A1
SCHEMBL3072114 0.71 PDE4B (0.52) MAOB
SCHEMBL3054495 0.71 PDE4B (0.52) SMN1; SMN2ALDH1A1KDM4EKMT2A
SCHEMBL6773687 0.70 NISCH (0.46) NISCHGAACLK4MAOBMAPT
SCHEMBL196765 0.70 CYP3A4 (0.73) NISCHGAADYRK1ACLK4MAOB
SCHEMBL29489425 0.70 CYP3A4 (0.73) NISCHGAADYRK1ACLK4MAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007047394-A2 THIOTRIAZOLYL DERIVATIVES EPIX DELAWARE, INC. (US) 2007-04-26 WO disclosed
WO-2007047394-A2 THIOTRIAZOLYL DERIVATIVES EPIX DELAWARE, INC. (US) 2007-04-26 WO disclosed