SCHEMBL5333231

SCHEMBL5333231

CC(C)C(N)C(=O)Nc1ccc(N2C(=O)N([C@@H](C)c3ccccc3)N=C(C3CCCCC3)c3ccccc32)cc1

nearest known ligand 0.74

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
PTH1R Q03431 12/20 0.74
CCKBR P32239 8/20 0.40
CCKAR P32238 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5333234 1.00 PTH1R (0.74) PTH1RCCKBRCCKAR
SCHEMBL5333228 1.00 PTH1R (0.74) PTH1RCCKBRCCKAR
SCHEMBL5329058 0.87 PTH1R (0.80) PTH1RCCKBRCCKAR
SCHEMBL5324433 0.86 PTH1R (0.74) PTH1RCCKBR
SCHEMBL14566324 0.85 PTH1R (1.00) PTH1RCCKBRCCKAR
SCHEMBL5322722 0.82 PTH1R (0.83) PTH1RCCKBRCCKAR
SCHEMBL5328766 0.81 PTH1R (0.77) PTH1RCCKBR
SCHEMBL5328774 0.81 PTH1R (0.77) PTH1RCCKBR
SCHEMBL5325329 0.81 PTH1R (0.81) PTH1RCCKBRCCKAR
SCHEMBL14566287 0.77 PTH1R (0.81) PTH1RCCKBRCCKAR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006129120-A9 BENZOTRIAZEPINONE DERIVATIVES JAMES BLACK FOUNDATION (GB) 2007-03-22 WO disclosed
WO-2006129120-A2 BENZOTRIAZEPINONE DERIVATIVES JAMES BLACK FOUNDATION (GB) 2006-12-07 WO disclosed