SCHEMBL5349191

SCHEMBL5349191

COC(=O)c1ccc2c(C3CCCCC3Br)c[nH]c2c1

nearest known ligand 0.49

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.49
ASH1L Q9NR48 1/20 0.43
KIF11 P52732 1/20 0.42
PARP1 P09874 2/20 0.40
GPR84 Q9NQS5 1/20 0.40
NR4A2 P43354 2/20 0.40
RAB9A P51151 1/20 0.39
HSD11B1 P28845 2/20 0.39
EIF2AK2 P19525 1/20 0.39
GSK3B P49841 1/20 0.39
ALDH1A1 P00352 2/20 0.38
MAPK1 P28482 1/20 0.38
HPGD P15428 1/20 0.38
PDE1C Q14123 1/20 0.38
ATM Q13315 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL391136 0.87 NPC1 (0.50) NPC1ASH1LKIF11PARP1GPR84
SCHEMBL391137 0.87 NPC1 (0.50) NPC1ASH1LKIF11PARP1GPR84
SCHEMBL391138 0.87 NPC1 (0.50) NPC1ASH1LKIF11PARP1GPR84
SCHEMBL393071 0.86 NPC1 (0.49) NPC1ASH1LKIF11PARP1GPR84
SCHEMBL393072 0.86 NPC1 (0.49) NPC1ASH1LKIF11PARP1GPR84
SCHEMBL393070 0.86 NPC1 (0.49) NPC1ASH1LKIF11PARP1GPR84
SCHEMBL1173868 0.84 NPC1 (0.54) NPC1ASH1LKIF11PARP1GPR84
SCHEMBL51234 0.83 NPC1 (0.53) NPC1ASH1LKIF11PARP1GPR84
SCHEMBL8877622 0.77 APP (0.54) NPC1ASH1LKIF11PARP1GPR84
SCHEMBL5447383 0.76 NPC1 (0.48) NPC1ASH1LKIF11PARP1GPR84

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007092000-A1 INHIBITORS OF HCV REPLICATION BRISTOL-MYERS SQUIBB COMPANY (US) 2007-08-16 WO disclosed