SCHEMBL5350832

SCHEMBL5350832

CCOc1cc(C2CNC(=O)C2)ccc1OC

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 20/20 1.00
PDE4B Q07343 14/20 0.80
PDE4C Q08493 14/20 0.80
PDE4D Q08499 14/20 0.80
CYP3A4 P08684 2/20 0.66
VEGFA P15692 1/20 0.66
ALDH1A1 P00352 1/20 0.66
LMNA P02545 1/20 0.66
CYP1A2 P05177 1/20 0.66
MAPT P10636 1/20 0.66
CYP2C9 P11712 1/20 0.66
ALOX15 P16050 1/20 0.66
CREBBP Q92793 1/20 0.66
KDM4E B2RXH2 1/20 0.66
PDE5A O76074 1/20 0.66
TNF P01375 1/20 0.66
MAPK1 P28482 1/20 0.66
BLM P54132 1/20 0.66
PDE1A P54750 1/20 0.66
PDE1B Q01064 1/20 0.66

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5326457 0.95 PDE4A (0.90) PDE4APDE4BPDE4CPDE4DCYP3A4
SCHEMBL5322466 0.93 PDE4A (0.87) PDE4APDE4BPDE4CPDE4DCYP3A4
SCHEMBL5329316 0.90 PDE4A (1.00) PDE4APDE4BPDE4CPDE4DCYP3A4
SCHEMBL7293719 0.89 PDE4A (1.00) PDE4APDE4BPDE4CPDE4DCYP3A4
SCHEMBL5324227 0.89 PDE4A (1.00) PDE4APDE4BPDE4CPDE4DCYP3A4
SCHEMBL5331581 0.88 PDE4A (0.79) PDE4APDE4BPDE4CPDE4DCYP3A4
SCHEMBL2790860 0.87 PDE4A (0.77) PDE4APDE4BPDE4CPDE4DCYP3A4
SCHEMBL2790858 0.87 PDE4A (0.77) PDE4APDE4BPDE4CPDE4DCYP3A4
SCHEMBL11486431 0.87 PDE4A (0.82) PDE4APDE4BPDE4CPDE4DCYP3A4
SCHEMBL5325679 0.87 PDE4A (0.91) PDE4APDE4BPDE4CPDE4DCYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4193926-A 4-(Polyalkoxy phenyl)-2-pyrrolidones SCHERING AKTIENGESELLSCHAFT (DE) 1980-03-18 US claimed
US-4012495-A USED IN TREATING NEUROLOGICAL AND PSYCHIC DISORDERS SCHERING AKTIENGESELLSCHAFT (DT) 1977-03-15 US claimed
WO-2007123699-A1 METHODS AND COMPOSITIONS FOR MODULATING MELANOGENESIS BY USING A MCLR AGONIST DANA-FARBER CANCER INSTITUTE, INC. (US) 2007-11-01 WO disclosed
US-4193926-A 4-(Polyalkoxy phenyl)-2-pyrrolidones SCHERING AKTIENGESELLSCHAFT (DE) 1980-03-18 US disclosed