SCHEMBL535471

SCHEMBL535471

CCOC(=O)CCCOc1cc(-c2noc(-c3ccc(-c4ccccc4C)c(COC)c3)n2)cc(F)c1F.COCc1cc(-c2nc(-c3cccc(COCCC(=O)OC(C)(C)C)c3)no2)ccc1-c1ccccc1C

nearest known ligand 0.51

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 19/20 0.51
S1PR3 Q99500 3/20 0.51
PTPN1 P18031 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL409995 0.88 S1PR1 (0.62) S1PR1S1PR3PTPN1
SCHEMBL410576 0.87 S1PR1 (0.60) S1PR1S1PR3
SCHEMBL2774789 0.83 S1PR1 (0.64) S1PR1S1PR3PTPN1
SCHEMBL410964 0.81 S1PR1 (0.67) S1PR1S1PR3
SCHEMBL2771037 0.78 S1PR1 (0.56) S1PR1S1PR3PTPN1
SCHEMBL407012 0.78 S1PR1 (0.70) S1PR1S1PR3
SCHEMBL2805557 0.76 S1PR1 (0.59) S1PR1S1PR3
SCHEMBL9968865 0.76 S1PR1 (0.63) S1PR1S1PR3
SCHEMBL409196 0.76 S1PR1 (0.57) S1PR1S1PR3
SCHEMBL13875177 0.76 S1PR1 (0.62) S1PR1S1PR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2414341-A2 OXADIAZOLE DERIVATIVES Merck Serono SA (CH) 2012-02-08 EP disclosed
WO-2010115751-A2 OXADIAZOLE DERIVATIVES MERCK SERONO S.A. (CH) 2010-10-14 WO disclosed