SCHEMBL5356295

SCHEMBL5356295

CN1CCN(S(=O)(=O)c2cc3cc(-c4cc5ccccc5[nH]c4=O)[nH]c3cc2F)CC1

nearest known ligand 0.73

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
KDR P35968 14/20 0.73
CHEK1 O14757 2/20 0.52
PKM P14618 1/20 0.39
VCP P55072 1/20 0.39
HRH4 Q9H3N8 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14590416 0.85 KDR (0.88) KDRCHEK1PKM
SCHEMBL5355012 0.85 KDR (1.00) KDRCHEK1PKM
SCHEMBL14590417 0.82 KDR (0.71) KDRCHEK1HRH4
SCHEMBL5356996 0.78 KDR (0.79) KDRPKMHRH4
SCHEMBL5357342 0.78 KDR (0.74) KDRCHEK1PKM
SCHEMBL14590415 0.74 KDR (0.55) KDRHRH4
SCHEMBL5371286 0.73 KDR (0.79) KDRHRH4
SCHEMBL5367396 0.73 KDR (1.00) KDRCHEK1PKM
SCHEMBL5357068 0.73 KDR (0.88) KDRCHEK1PKM
SCHEMBL5355475 0.73 KDR (0.68) KDRPKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7169788-B2 Tyrosine kinase inhibitors MERCK & CO., INC. (US) 2007-01-30 US disclosed
US-7169788-B2 Tyrosine kinase inhibitors MERCK & CO., INC. (US) 2007-01-30 US disclosed
US-7169788-B2 Tyrosine kinase inhibitors MERCK & CO., INC. (US) 2007-01-30 US disclosed