SCHEMBL5357450

SCHEMBL5357450

O=C(O)c1cc(Cl)ccc1Oc1cncc(F)c1

nearest known ligand 0.54

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
EPAS1 Q99814 1/20 0.48
PTGER4 P35408 4/20 0.47
GRM5 P41594 1/20 0.46
XDH P47989 3/20 0.45
SLC22A12 Q96S37 2/20 0.45
PTGER2 P43116 2/20 0.44
GAA P10253 2/20 0.44
TSHR P16473 1/20 0.44
CYP3A4 P08684 2/20 0.43
VEGFA P15692 1/20 0.43
ALDH1A1 P00352 1/20 0.42
POLB P06746 1/20 0.42
HPGD P15428 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5357696 0.87 PPARG (0.52) PTGER4XDHSLC22A12GAATSHR
SCHEMBL5364950 0.86 EPAS1 (0.51) EPAS1PTGER4GRM5PTGER2CYP3A4
SCHEMBL5363227 0.84 EPAS1 (0.60) EPAS1PTGER4PTGER2GAATSHR
SCHEMBL4448975 0.81 PTGER4 (0.62) EPAS1PTGER4PTGER2GAATSHR
SCHEMBL4447285 0.81 PTGER4 (0.62) EPAS1PTGER4PTGER2GAATSHR
SCHEMBL5817933 0.81 PTGER4 (0.42) EPAS1PTGER4GRM5XDHSLC22A12
SCHEMBL5365760 0.79 PTGER4 (0.77) PTGER4PTGER2
SCHEMBL3981747 0.79 NR4A2 (0.47) PTGER4
SCHEMBL11577659 0.78 GAA (0.54) PTGER4PTGER2GAATSHRALDH1A1
SCHEMBL5357266 0.77 GAA (0.51) EPAS1PTGER4PTGER2GAATSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1663979-B1 PHENYL OR PYRIDYL AMIDE COMPOUNDS AS PROSTAGLANDIN E2 ANTAGONISTS RAQUALIA PHARMA INC (JP) 2013-10-09 EP disclosed
US-7238714-B2 Aryl or heteroaryl amide compounds PFIZER JAPAN, INC. (JP) 2007-07-03 US disclosed
EP-1663979-A1 PHENYL OR PYRIDYL AMIDE COMPOUNDS AS PROSTAGLANDIN E2 ANTAGONISTS PFIZER INC. (US) 2006-06-07 EP disclosed
US-20050065188-A1 Aryl or heteroaryl amide compounds ASKAT INC. (JP) 2005-03-24 US disclosed
WO-2005021508-A1 PHENYL OR PYRIDYL AMIDE COMPOUNDS AS PROSTAGLANDIN E2 ANTAGONISTS PFIZER INC. (US) 2005-03-10 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050065188-A1 Aryl or heteroaryl amide compounds HRH2, PTGER1, LTB4R2 EPAS1 1007/4885PTGER4 13/4885GRM5 787/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.