SCHEMBL536168

SCHEMBL536168

C[C@@H]1CCCCN1c1ccc(C(=O)O)cc1C(F)(F)F.C[C@H]1CCCCN1c1ccc(C(=O)O)cc1C(F)(F)F

nearest known ligand 0.49

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 7/20 0.49
GPBAR1 Q8TDU6 1/20 0.48
GFER P55789 1/20 0.48
TTR P02766 1/20 0.44
TAS1R3 Q7RTX0 1/20 0.43
TAS1R1 Q7RTX1 1/20 0.43
TAS1R2 Q8TE23 1/20 0.43
GAA P10253 2/20 0.43
HPGD P15428 1/20 0.43
RARA P10276 1/20 0.42
RARB P10826 1/20 0.42
RARG P13631 1/20 0.42
KDM4E B2RXH2 1/20 0.42
POLB P06746 1/20 0.42
NR4A1 P22736 1/20 0.42
HSD17B10 Q99714 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL409116 1.00 S1PR1 (0.49) S1PR1GPBAR1GFERTTRTAS1R3
SCHEMBL405390 1.00 S1PR1 (0.49) S1PR1GPBAR1GFERTTRTAS1R3
SCHEMBL410127 1.00 S1PR1 (0.49) S1PR1GPBAR1GFERTTRTAS1R3
Hydrochloric Acid SCHEMBL2810962 0.99 S1PR1 (0.48) S1PR1GPBAR1GFERTTRTAS1R3
SCHEMBL2484886 0.92 S1PR1 (0.52) S1PR1GPBAR1GFERTTRRARA
SCHEMBL18373542 0.91 GFER (0.47) S1PR1GPBAR1GFERTTRGAA
SCHEMBL1725667 0.88 S1PR1 (0.48) S1PR1GPBAR1GFERTTRRARA
SCHEMBL410194 0.87 S1PR1 (0.50) S1PR1GPBAR1GFERGAAHPGD
Hydrochloric Acid SCHEMBL16817128 0.86 S1PR1 (0.49) S1PR1GPBAR1GFERGAAHPGD
SCHEMBL20702699 0.82 S1PR1 (0.48) S1PR1GPBAR1GFERGAAHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2414342-A1 OXADIAZOLE DERIVATIVES Merck Serono S.A. (CH) 2012-02-08 EP disclosed