SCHEMBL5363069

SCHEMBL5363069

CNS(=O)(=O)c1ccc2c(c1)C(=Cc1ccc(O)c(C(C)(C)C)c1)C(=O)N2

nearest known ligand 0.51

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
SRC P12931 2/20 0.51
ERBB2 P04626 3/20 0.50
EGFR P00533 2/20 0.50
IGF1R P08069 1/20 0.50
CDK2 P24941 2/20 0.49
PLK4 O00444 1/20 0.48
KDR P35968 1/20 0.48
NOX4 Q9NPH5 1/20 0.47
NTRK1 P04629 1/20 0.47
FCER2 P06734 1/20 0.47
SYK P43405 1/20 0.47
NTRK3 Q16288 1/20 0.47
NTRK2 Q16620 1/20 0.47
AURKA O14965 1/20 0.46
LRRK2 Q5S007 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5365058 0.90 ERBB2 (0.64) SRCERBB2EGFRIGF1RCDK2
SCHEMBL5363044 0.86 SRC (0.53) SRCCDK2PLK4KDRNOX4
SCHEMBL5367619 0.86 ERBB2 (0.68) SRCERBB2EGFRIGF1RCDK2
SCHEMBL5369480 0.86 ERBB2 (0.56) SRCERBB2EGFRIGF1RCDK2
SCHEMBL5358229 0.85 LRRK2 (0.64) SRCEGFRCDK2PLK4KDR
SCHEMBL5365593 0.85 ERBB2 (0.55) SRCERBB2EGFRIGF1RCDK2
SCHEMBL5359293 0.85 RAF1 (0.55) SRCERBB2EGFRIGF1RCDK2
SCHEMBL5367175 0.84 MOGAT2 (0.53) ERBB2EGFRIGF1RPLK4NOX4
SCHEMBL7135152 0.84 SRC (0.55) SRCCDK2KDRNTRK1FCER2
SCHEMBL5365190 0.84 PSEN1 (0.60) SRCCDK2PLK4KDRLRRK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7202265-B2 Indolinone combinatorial libraries and related products and methods for the treatment of disease SUGEN, INC. (US) 2007-04-10 US disclosed
US-20050197382-A1 Indolinone combinatorial libraries and related products and methods for the treatment of disease SUGEN, INC. 2005-09-08 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050197382-A1 Indolinone combinatorial libraries and related products and methods for the treatment of disease FRK, PTK2, DSTYK SRC 189/4885ERBB2 19/4885EGFR 286/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.