SCHEMBL5365601

SCHEMBL5365601

Cc1ccsc1C=C1C(=O)Nc2ccc(CCCl)cc21

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 5/20 0.45
KMT2A Q03164 5/20 0.45
KDR P35968 2/20 0.44
ALDH1A1 P00352 4/20 0.43
MAPT P10636 4/20 0.43
NPC1 O15118 3/20 0.43
RAB9A P51151 1/20 0.43
S1PR4 O95977 1/20 0.42
HSP90AA1 P07900 1/20 0.42
ALOX12 P18054 1/20 0.42
S1PR1 P21453 1/20 0.42
NTSR1 P30989 1/20 0.42
HTT P42858 1/20 0.42
NPSR1 Q6W5P4 1/20 0.42
TDP1 Q9NUW8 1/20 0.42
RET P07949 4/20 0.41
LRRK2 Q5S007 2/20 0.41
POLB P06746 1/20 0.41
PDPK1 O15530 3/20 0.41
PDGFRB P09619 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5374098 0.86 KDR (0.61) MEN1KMT2AKDRALDH1A1MAPT
SCHEMBL5364110 0.86 PDPK1 (0.56) MEN1KMT2AKDRALDH1A1MAPT
SCHEMBL5358278 0.86 MEN1 (0.46) MEN1KMT2AKDRALDH1A1MAPT
SCHEMBL6297819 0.82 LRRK2 (0.60) RETLRRK2PDGFRB
SCHEMBL6297823 0.82 LRRK2 (0.60) RETLRRK2PDGFRB
SCHEMBL7133841 0.81 MEN1 (0.59) MEN1KMT2AKDRALDH1A1MAPT
SCHEMBL5363153 0.80 RET (0.37) MEN1KMT2AKDRALDH1A1MAPT
SCHEMBL5357949 0.80 RET (0.41) MEN1KMT2AKDRRETLRRK2
SCHEMBL7139419 0.79 MEN1 (0.67) MEN1KMT2AKDRMAPTNPC1
SCHEMBL7137564 0.79 PSEN1 (0.52) MEN1KMT2AMAPTRETLRRK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7202265-B2 Indolinone combinatorial libraries and related products and methods for the treatment of disease SUGEN, INC. (US) 2007-04-10 US disclosed
US-20050197382-A1 Indolinone combinatorial libraries and related products and methods for the treatment of disease SUGEN, INC. 2005-09-08 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050197382-A1 Indolinone combinatorial libraries and related products and methods for the treatment of disease FRK, PTK2, DSTYK MEN1 3855/4885KMT2A 4060/4885KDR 239/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.