SCHEMBL5366100

SCHEMBL5366100

COC(=O)c1cc(Cl)ccc1Cc1cccc(F)c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.47
ALDH1A1 P00352 1/20 0.47
HPGD P15428 1/20 0.47
MAPK1 P28482 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
HSD17B10 Q99714 1/20 0.47
L3MBTL1 Q9Y468 1/20 0.47
SNCA P37840 6/20 0.45
PLA2G2A P14555 2/20 0.45
HSP90AA1 P07900 1/20 0.44
ABL1 P00519 1/20 0.43
MRGPRX4 Q96LA9 1/20 0.43
KMT2A Q03164 2/20 0.43
PPARG P37231 2/20 0.43
PPARA Q07869 2/20 0.43
MEN1 O00255 1/20 0.43
IDE P14735 1/20 0.43
MAOA P21397 1/20 0.43
MAOB P27338 1/20 0.43
CNR1 P21554 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5365504 0.89 HSP90AA1 (0.53) KDM4EALDH1A1HPGDMAPK1HSD17B10
SCHEMBL5357513 0.84 PPARG (0.46) ALDH1A1HPGDHSD17B10SNCAMRGPRX4
SCHEMBL5367029 0.81 PTGER4 (0.57) ALDH1A1
SCHEMBL3980074 0.81 MRGPRX4 (0.57) ABL1MRGPRX4MAOAMAOBNR4A2
SCHEMBL4450367 0.79 KDM4E (0.49) KDM4EALDH1A1HPGDMAPK1SMN1; SMN2
SCHEMBL9937243 0.76 MRGPRX4 (0.54) KDM4EALDH1A1HPGDMAPK1SMN1; SMN2
SCHEMBL9938816 0.76 MAOB (0.50) KDM4EALDH1A1HPGDMAPK1SMN1; SMN2
SCHEMBL10174510 0.76 ABL1 (0.57) KDM4EALDH1A1HPGDMAPK1PLA2G2A
SCHEMBL3980720 0.74 FABP3 (0.45) SMN1; SMN2L3MBTL1ABL1MRGPRX4KMT2A
SCHEMBL4768171 0.74 IDO1 (0.44) HPGDMAPK1SMN1; SMN2HSD17B10L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1663979-B1 PHENYL OR PYRIDYL AMIDE COMPOUNDS AS PROSTAGLANDIN E2 ANTAGONISTS RAQUALIA PHARMA INC (JP) 2013-10-09 EP disclosed
CN-1867551-B Phenyl or pyridyl amide compounds as prostaglandin E2 antagonists RAQUALIA PHARMA INC 2013-09-11 CN disclosed
US-7238714-B2 Aryl or heteroaryl amide compounds PFIZER JAPAN, INC. (JP) 2007-07-03 US disclosed
CN-1867551-A Phenyl or pyridyl amide compounds as prostaglandin E2 antagonists PFIZER (US) 2006-11-22 CN disclosed
EP-1663979-A1 PHENYL OR PYRIDYL AMIDE COMPOUNDS AS PROSTAGLANDIN E2 ANTAGONISTS PFIZER INC. (US) 2006-06-07 EP disclosed
US-20050065188-A1 Aryl or heteroaryl amide compounds ASKAT INC. (JP) 2005-03-24 US disclosed
WO-2005021508-A1 PHENYL OR PYRIDYL AMIDE COMPOUNDS AS PROSTAGLANDIN E2 ANTAGONISTS PFIZER INC. (US) 2005-03-10 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050065188-A1 Aryl or heteroaryl amide compounds HRH2, PTGER1, LTB4R2 KDM4E 875/4885ALDH1A1 860/4885HPGD 215/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.