SCHEMBL5366152

SCHEMBL5366152

Cc1ccsc1C=C1C(=O)Nc2ccc(C(=O)Nc3ccccc3)cc21

nearest known ligand 0.51

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 3/20 0.51
TLK2 Q86UE8 6/20 0.51
JAK3 P52333 3/20 0.50
PAK4 O96013 3/20 0.49
KDR P35968 2/20 0.47
EGFR P00533 1/20 0.47
PDGFRB P09619 1/20 0.47
FGFR1 P11362 1/20 0.47
RET P07949 1/20 0.44
NTRK1 P04629 1/20 0.44
TP53 P04637 1/20 0.44
MAPT P10636 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5367344 0.85 GRK5 (0.51) GSK3BJAK3PAK4KDREGFR
SCHEMBL5366782 0.82 PDPK1 (0.60) TLK2JAK3KDRMAPT
SCHEMBL5366834 0.81 GSK3B (0.52) GSK3BTLK2JAK3PAK4KDR
SCHEMBL5361474 0.81 TLK2 (0.70) TLK2JAK3PAK4KDREGFR
SCHEMBL13712838 0.81 GSK3B (0.55) GSK3BTLK2JAK3KDREGFR
SCHEMBL5364206 0.80 JAK3 (0.47) TLK2JAK3PAK4KDRMAPT
SCHEMBL5361229 0.79 AKT2 (0.59) GSK3B
SCHEMBL5359359 0.79 TLK2 (0.47) TLK2JAK3KDRRETMAPT
SCHEMBL5362148 0.78 KDR (0.48) GSK3BTLK2JAK3KDRPDGFRB
SCHEMBL5363197 0.77 TLK2 (0.80) TLK2JAK3PAK4PDGFRBNTRK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7202265-B2 Indolinone combinatorial libraries and related products and methods for the treatment of disease SUGEN, INC. (US) 2007-04-10 US disclosed
US-20050197382-A1 Indolinone combinatorial libraries and related products and methods for the treatment of disease SUGEN, INC. 2005-09-08 US disclosed
EP-1247803-A2 Indolinone compounds suitable for modulation of protein kinases Sugen, Inc. (US) 2002-10-09 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050197382-A1 Indolinone combinatorial libraries and related products and methods for the treatment of disease FRK, PTK2, DSTYK GSK3B 315/4885TLK2 48/4885JAK3 40/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.