SCHEMBL5367067

SCHEMBL5367067

Cc1cc(Br)cc(Oc2cc(Cc3ccc(=O)[nH]n3)ccc2Cl)c1

nearest known ligand 0.43

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 4/20 0.43
THRA P10827 1/20 0.34
THRB P10828 1/20 0.34
KDM4E B2RXH2 1/20 0.32
NPC1 O15118 1/20 0.32
RAB9A P51151 1/20 0.32
HTR2A P28223 1/20 0.31
SLC6A4 P31645 1/20 0.31
KCNH2 Q12809 1/20 0.31
CYP2C9 P11712 1/20 0.30
CYP2C19 P33261 1/20 0.30
SMN1; SMN2 Q16637 1/20 0.30
ADORA2A P29274 1/20 0.30
ADORA1 P30542 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5381986 0.92 CYP3A4 (0.47) CYP3A4THRATHRBKDM4ENPC1
SCHEMBL5373776 0.88 CYP3A4 (0.43) CYP3A4THRATHRBCYP2C9CYP2C19
SCHEMBL5375943 0.87 CYP3A4 (0.42) CYP3A4THRATHRBHTR2ASLC6A4
SCHEMBL5366918 0.86 CYP3A4 (0.47) CYP3A4THRATHRBHTR2ASLC6A4
SCHEMBL5364926 0.85 CYP3A4 (0.54) CYP3A4THRATHRBRAB9AHTR2A
SCHEMBL5385784 0.85 CYP3A4 (0.44) CYP3A4THRATHRBKDM4ENPC1
SCHEMBL5368714 0.83 CYP3A4 (0.53) CYP3A4THRATHRBKDM4ENPC1
SCHEMBL5381993 0.81 CYP3A4 (0.47) CYP3A4THRATHRBKDM4ENPC1
SCHEMBL5373613 0.81 CYP3A4 (0.51) CYP3A4THRATHRBHTR2ASLC6A4
SCHEMBL4367667 0.81 CYP3A4 (0.53) CYP3A4THRATHRBCYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7189718-B2 Non-nucleoside reverse transcriptase inhibitors ROCHE PALO ALTO LLC (US) 2007-03-13 US disclosed
US-7189718-B2 Non-nucleoside reverse transcriptase inhibitors ROCHE PALO ALTO LLC (US) 2007-03-13 US disclosed
US-7189718-B2 Non-nucleoside reverse transcriptase inhibitors ROCHE PALO ALTO LLC (US) 2007-03-13 US disclosed