SCHEMBL5367150

SCHEMBL5367150

CC(C)(C)c1cc(C=C2C(=O)Nc3ccc(I)cc32)cc(Cl)c1O

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAF1 P04049 6/20 0.61
EGFR P00533 4/20 0.61
ERBB2 P04626 4/20 0.61
MAPT P10636 3/20 0.61
MAP1LC3B Q9GZQ8 2/20 0.61
PLK4 O00444 2/20 0.61
PLK1 P53350 2/20 0.61
KIF15 Q9NS87 2/20 0.61
NTRK1 P04629 1/20 0.61
ARAF P10398 1/20 0.61
PIM1 P11309 1/20 0.61
BRAF P15056 1/20 0.61
CSNK2A1 P68400 1/20 0.61
PIM3 Q86V86 1/20 0.61
SIRT2 Q8IXJ6 1/20 0.61
SIRT1 Q96EB6 1/20 0.61
MYOC Q99972 1/20 0.61
DYRK4 Q9NR20 1/20 0.61
SIRT3 Q9NTG7 1/20 0.61
SIRT5 Q9NXA8 1/20 0.61

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5361193 0.88 ERBB2 (0.63) RAF1EGFRERBB2MAPTMAP1LC3B
SCHEMBL5367163 0.87 RAF1 (0.79) RAF1EGFRERBB2MAPTMAP1LC3B
SCHEMBL5368201 0.85 ERBB2 (0.66) RAF1EGFRERBB2MAPTMAP1LC3B
SCHEMBL5366594 0.83 ERBB2 (0.57) RAF1EGFRERBB2MAP1LC3BPLK4
SCHEMBL5468784 0.83 LRRK2 (0.72) EGFRERBB2IGF1RLRRK2PSEN1
SCHEMBL5468785 0.83 LRRK2 (0.72) EGFRERBB2IGF1RLRRK2PSEN1
SCHEMBL5365593 0.82 ERBB2 (0.55) RAF1EGFRERBB2PLK4PLK1
SCHEMBL6690796 0.81 RAF1 (0.76) RAF1EGFRERBB2MAPTMAP1LC3B
SCHEMBL5358336 0.80 ERBB2 (0.52) RAF1EGFRERBB2MAPTMAP1LC3B
SCHEMBL7319104 0.79 ERBB2 (0.73) RAF1EGFRERBB2MAPTMAP1LC3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7202265-B2 Indolinone combinatorial libraries and related products and methods for the treatment of disease SUGEN, INC. (US) 2007-04-10 US disclosed
US-20050197382-A1 Indolinone combinatorial libraries and related products and methods for the treatment of disease SUGEN, INC. 2005-09-08 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050197382-A1 Indolinone combinatorial libraries and related products and methods for the treatment of disease FRK, PTK2, DSTYK RAF1 245/4885EGFR 286/4885ERBB2 19/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.