SCHEMBL5368441

SCHEMBL5368441

N#Cc1ccc(Oc2c(Cl)ccc(Cc3ccc(=O)[nH]n3)c2F)cc1

nearest known ligand 0.58

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 4/20 0.58
CYP2C9 P11712 1/20 0.58
CYP2C19 P33261 1/20 0.58
PGR P06401 3/20 0.37
THRA P10827 2/20 0.35
THRB P10828 2/20 0.35
HTR2A P28223 2/20 0.34
KCNH2 Q12809 2/20 0.34
MERTK Q12866 1/20 0.33
SLC6A4 P31645 1/20 0.32
AKR1B1 P15121 1/20 0.32
PRMT5 O14744 1/20 0.32
WDR77 Q9BQA1 1/20 0.32
EPHX2 P34913 1/20 0.32
CYP11B1 P15538 2/20 0.32
CYP11B2 P19099 1/20 0.32
KDR P35968 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5368884 0.91 CYP3A4 (0.68) CYP3A4CYP2C9CYP2C19THRATHRB
SCHEMBL14570716 0.88 CYP3A4 (0.60) CYP3A4CYP2C9CYP2C19THRATHRB
SCHEMBL14559741 0.88 CYP3A4 (0.75) CYP3A4CYP2C9CYP2C19THRATHRB
SCHEMBL5373843 0.88 CYP3A4 (0.65) CYP3A4CYP2C9CYP2C19THRATHRB
SCHEMBL5364946 0.88 CYP3A4 (0.54) CYP3A4CYP2C9CYP2C19THRATHRB
SCHEMBL5373271 0.86 CYP3A4 (0.68) CYP3A4CYP2C9CYP2C19THRATHRB
SCHEMBL5367059 0.86 CYP3A4 (0.48) CYP3A4CYP2C9CYP2C19THRATHRB
SCHEMBL5367044 0.85 CYP3A4 (0.52) CYP3A4CYP2C9CYP2C19THRATHRB
SCHEMBL5331103 0.85 CYP3A4 (0.61) CYP3A4CYP2C9CYP2C19THRATHRB
SCHEMBL5373625 0.85 CYP3A4 (0.63) CYP3A4CYP2C9CYP2C19PGRTHRA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7189718-B2 Non-nucleoside reverse transcriptase inhibitors ROCHE PALO ALTO LLC (US) 2007-03-13 US disclosed
US-7189718-B2 Non-nucleoside reverse transcriptase inhibitors ROCHE PALO ALTO LLC (US) 2007-03-13 US disclosed