SCHEMBL5368624

SCHEMBL5368624

Cc1cc(Cc2ccc(Cl)c(Oc3cccc(C#N)c3)c2F)n[nH]c1=O

nearest known ligand 0.80

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 3/20 0.80
CYP2C9 P11712 1/20 0.80
CYP2C19 P33261 1/20 0.80
SLC5A2 P31639 1/20 0.39
PRMT5 O14744 1/20 0.38
WDR77 Q9BQA1 1/20 0.38
KCNH2 Q12809 4/20 0.35
HTR2A P28223 3/20 0.35
NPBWR1 P48145 1/20 0.35
MCHR1 Q99705 1/20 0.35
PIK3R1 P27986 2/20 0.33
PIK3CA P42336 2/20 0.33
SLC6A4 P31645 2/20 0.33
EPHX2 P34913 1/20 0.33
P2RX3 P56373 1/20 0.33
EPAS1 Q99814 3/20 0.32
BCAT2 O15382 1/20 0.32
BCAT1 P54687 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4274657 0.92 CYP3A4 (0.91) CYP3A4CYP2C9CYP2C19SLC5A2KCNH2
SCHEMBL5370521 0.92 CYP3A4 (0.67) CYP3A4CYP2C9CYP2C19SLC5A2PRMT5
SCHEMBL5370387 0.90 CYP3A4 (0.65) CYP3A4CYP2C9CYP2C19SLC5A2PRMT5
SCHEMBL4272969 0.89 CYP3A4 (1.00) CYP3A4CYP2C9CYP2C19SLC5A2KCNH2
SCHEMBL5368425 0.89 CYP3A4 (0.86) CYP3A4CYP2C9CYP2C19SLC5A2KCNH2
SCHEMBL5374302 0.89 CYP3A4 (0.64) CYP3A4CYP2C9CYP2C19SLC5A2PRMT5
SCHEMBL4274479 0.89 CYP3A4 (0.86) CYP3A4CYP2C9CYP2C19SLC5A2KCNH2
SCHEMBL5374165 0.87 CYP3A4 (0.74) CYP3A4CYP2C9CYP2C19SLC5A2KCNH2
SCHEMBL5368877 0.86 CYP3A4 (0.70) CYP3A4CYP2C9CYP2C19SLC5A2NPBWR1
SCHEMBL5344677 0.86 CYP3A4 (0.81) CYP3A4CYP2C9CYP2C19SLC5A2KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7189718-B2 Non-nucleoside reverse transcriptase inhibitors ROCHE PALO ALTO LLC (US) 2007-03-13 US disclosed