SCHEMBL5369959

SCHEMBL5369959

CCCN(CCC)C(=O)c1cc(C)cc(C(=O)N[C@@H](Cc2cc(F)cc(F)c2)[C@H](O)CNC[C@H](C)CC)c1

nearest known ligand 0.75

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 20/20 0.75
BACE2 Q9Y5Z0 5/20 0.75
CTSD P07339 3/20 0.72

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3354903 0.93 BACE1 (0.78) BACE1BACE2CTSD
SCHEMBL3352358 0.93 BACE1 (0.78) BACE1BACE2CTSD
SCHEMBL5378355 0.93 BACE1 (0.78) BACE1BACE2CTSD
SCHEMBL3348995 0.93 BACE1 (0.78) BACE1BACE2CTSD
SCHEMBL3354515 0.91 BACE1 (0.80) BACE1BACE2CTSD
SCHEMBL5348605 0.90 BACE1 (0.88) BACE1BACE2CTSD
SCHEMBL3348915 0.89 BACE1 (0.75) BACE1BACE2CTSD
SCHEMBL5354471 0.89 BACE1 (0.87) BACE1BACE2CTSD
SCHEMBL5363946 0.89 BACE1 (0.74) BACE1BACE2CTSD
SCHEMBL8356578 0.89 BACE1 (0.72) BACE1BACE2CTSD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7176242-B2 N,N′-substituted-1,3-diamino-2-hydroxypropane derivatives ELAN PHARMACEUTICALS, INC. (US) 2007-02-13 US claimed