SCHEMBL5370108

SCHEMBL5370108

CN(C1CCNC1)S(=O)(=O)c1ccc2[nH]c(-c3cc4c(F)cccc4[nH]c3=O)cc2c1

nearest known ligand 0.52

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
SLC6A2 P23975 3/20 0.52
SLC6A4 P31645 3/20 0.52
KDR P35968 8/20 0.51
KCNH2 Q12809 1/20 0.37
CHEK1 O14757 2/20 0.36
MAPT P10636 1/20 0.35
DAO P14920 1/20 0.34
DDO Q99489 1/20 0.34
ALOX5AP P20292 3/20 0.34
FEN1 P39748 3/20 0.34
FLT3 P36888 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5354782 0.88 KDR (0.65) SLC6A2SLC6A4KDRKCNH2CHEK1
SCHEMBL5370412 0.82 SLC6A2 (0.62) SLC6A2SLC6A4KDRKCNH2CHEK1
SCHEMBL5371327 0.79 SLC6A2 (0.56) SLC6A2SLC6A4KDRKCNH2MAPT
SCHEMBL5361067 0.79 KDR (0.49) SLC6A2SLC6A4KDRCHEK1ALOX5AP
SCHEMBL5354528 0.78 KDR (0.50) SLC6A2SLC6A4KDRCHEK1ALOX5AP
SCHEMBL5350566 0.76 SLC6A2 (0.56) SLC6A2SLC6A4KDRKCNH2ALOX5AP
SCHEMBL5362169 0.72 KDR (0.77) KDRCHEK1ALOX5APFEN1
SCHEMBL5363140 0.69 KDR (0.63) KDRCHEK1
SCHEMBL143284 0.68 KDR (0.65) SLC6A2SLC6A4KDRKCNH2CHEK1
SCHEMBL5355525 0.68 KDR (1.00) KDRCHEK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7169788-B2 Tyrosine kinase inhibitors MERCK & CO., INC. (US) 2007-01-30 US disclosed
US-7169788-B2 Tyrosine kinase inhibitors MERCK & CO., INC. (US) 2007-01-30 US disclosed
US-7169788-B2 Tyrosine kinase inhibitors MERCK & CO., INC. (US) 2007-01-30 US disclosed