SCHEMBL5370180

SCHEMBL5370180

Cc1ccc(C#N)cc1Oc1c(C)ccc(Cc2cc(C)c(=O)[nH]n2)c1F

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 3/20 0.61
CYP2C9 P11712 1/20 0.61
CYP2C19 P33261 1/20 0.61
CHRM2 P08172 1/20 0.33
CHRM1 P11229 1/20 0.33
RRM1 P23921 1/20 0.33
RRM2B Q7LG56 1/20 0.33
SLC5A2 P31639 1/20 0.33
AR P10275 2/20 0.32
HTR2A P28223 1/20 0.31
KCNH2 Q12809 1/20 0.31
DRD1 P21728 1/20 0.31
FFAR1 O14842 1/20 0.31
FFAR4 Q5NUL3 1/20 0.31
SCN8A Q9UQD0 1/20 0.30
SCN10A Q9Y5Y9 1/20 0.30
PIK3R1 P27986 1/20 0.30
PIK3CA P42336 1/20 0.30
PTGDR2 Q9Y5Y4 1/20 0.30
LRRK2 Q5S007 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14570777 0.92 CYP3A4 (0.58) CYP3A4CYP2C9CYP2C19CHRM2CHRM1
SCHEMBL5377154 0.92 CYP3A4 (0.68) CYP3A4CYP2C9CYP2C19CHRM2CHRM1
SCHEMBL5366810 0.88 CYP3A4 (0.49) CYP3A4CYP2C9CYP2C19CHRM2CHRM1
SCHEMBL5374165 0.87 CYP3A4 (0.74) CYP3A4CYP2C9CYP2C19CHRM2CHRM1
SCHEMBL5668069 0.87 CYP3A4 (0.76) CYP3A4CYP2C9CYP2C19SLC5A2KCNH2
SCHEMBL5370521 0.86 CYP3A4 (0.67) CYP3A4CYP2C9CYP2C19SLC5A2AR
SCHEMBL5377646 0.86 CYP3A4 (0.67) CYP3A4CYP2C9CYP2C19SLC5A2AR
SCHEMBL5376896 0.84 CYP3A4 (0.65) CYP3A4CYP2C9CYP2C19SLC5A2AR
SCHEMBL5375519 0.83 CYP3A4 (0.76) CYP3A4CYP2C9CYP2C19SLC5A2HTR2A
SCHEMBL5377555 0.81 CYP3A4 (0.54) CYP3A4CYP2C9CYP2C19CHRM2CHRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7189718-B2 Non-nucleoside reverse transcriptase inhibitors ROCHE PALO ALTO LLC (US) 2007-03-13 US disclosed
US-7189718-B2 Non-nucleoside reverse transcriptase inhibitors ROCHE PALO ALTO LLC (US) 2007-03-13 US disclosed
US-7189718-B2 Non-nucleoside reverse transcriptase inhibitors ROCHE PALO ALTO LLC (US) 2007-03-13 US disclosed