SCHEMBL5370753

SCHEMBL5370753

CCc1cccc(CNC[C@H](O)[C@H](Cc2cc(F)cc(F)c2)NC(=O)c2cc(C)cc(C(=O)O)c2)c1

nearest known ligand 0.79

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 20/20 0.79
CTSD P07339 2/20 0.79
BACE2 Q9Y5Z0 3/20 0.69
CTSB P07858 7/20 0.63

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5370751 1.00 BACE1 (0.79) BACE1CTSDBACE2CTSB
Hydrochloric Acid SCHEMBL3349144 0.99 BACE1 (0.77) BACE1CTSDBACE2CTSB
Hydrochloric Acid SCHEMBL3349138 0.99 BACE1 (0.77) BACE1CTSDBACE2CTSB
SCHEMBL3356940 0.95 BACE1 (0.82) BACE1CTSDBACE2CTSB
SCHEMBL3356941 0.95 BACE1 (0.82) BACE1CTSDBACE2CTSB
SCHEMBL13306778 0.95 BACE1 (0.82) BACE1CTSDBACE2CTSB
SCHEMBL3383926 0.93 BACE1 (0.76) BACE1CTSDBACE2CTSB
SCHEMBL3350448 0.93 BACE1 (0.76) BACE1CTSDBACE2CTSB
SCHEMBL5353188 0.93 BACE1 (0.76) BACE1CTSDBACE2CTSB
SCHEMBL7612911 0.93 BACE1 (0.79) BACE1CTSDBACE2CTSB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7176242-B2 N,N′-substituted-1,3-diamino-2-hydroxypropane derivatives ELAN PHARMACEUTICALS, INC. (US) 2007-02-13 US claimed
EP-1453789-A2 N,N'-SUBSTITUTED-1,3-DIAMINO-2-HYDROXYPROPANE DERIVATIVES Elan Pharmaceuticals, Inc. (US) 2004-09-08 EP claimed
WO-2003040096-A2 N, N'-SUBSTITUTED-1,3-DIAMINO-2-HYDROXYPROPANE DERIVATIVES ELAN PHARMACEUTICALS, INC. (US) 2003-05-15 WO claimed