SCHEMBL5373428

SCHEMBL5373428

CCCN(CCC)C(=O)c1cccc(C(N)=O)c1[C@H](Cc1ccccc1)[C@@H](O)CNCc1ccccc1OC(F)(F)F

nearest known ligand 0.43

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 15/20 0.43
CTSD P07339 9/20 0.43
BCHE P06276 3/20 0.41
PPARG P37231 2/20 0.41
EPHX2 P34913 1/20 0.38
BACE2 Q9Y5Z0 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3347371 0.87 BACE1 (0.45) BACE1CTSDBACE2
SCHEMBL3351421 0.86 BACE1 (0.47) BACE1CTSDBACE2
SCHEMBL3349771 0.86 BACE1 (0.45) BACE1CTSDBACE2
SCHEMBL3348139 0.85 BACE1 (0.43) BACE1CTSDBACE2
SCHEMBL3351487 0.85 BACE1 (0.45) BACE1CTSDBACE2
SCHEMBL3351399 0.84 BACE1 (0.44) BACE1CTSDBACE2
SCHEMBL3351667 0.84 BACE1 (0.44) BACE1CTSDBACE2
SCHEMBL3350577 0.84 BACE1 (0.43) BACE1CTSDBACE2
SCHEMBL3348246 0.83 BACE1 (0.53) BACE1CTSDBCHE
SCHEMBL3349119 0.83 BACE1 (0.46) BACE1CTSDBCHEBACE2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7176242-B2 N,N′-substituted-1,3-diamino-2-hydroxypropane derivatives ELAN PHARMACEUTICALS, INC. (US) 2007-02-13 US disclosed