SCHEMBL5374665

SCHEMBL5374665

CCc1cccc(CNC[C@H](O)[C@@H](Cc2cc(F)cc(F)c2)NC(=O)c2cccc(C(=O)C(C)C)c2)c1

nearest known ligand 0.68

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 20/20 0.68
CTSD P07339 3/20 0.68
CTSB P07858 4/20 0.60
BACE2 Q9Y5Z0 2/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5374658 1.00 BACE1 (0.68) BACE1CTSDCTSBBACE2
SCHEMBL3352084 0.92 BACE1 (0.67) BACE1CTSDCTSBBACE2
SCHEMBL3352079 0.92 BACE1 (0.67) BACE1CTSDCTSBBACE2
Hydrochloric Acid SCHEMBL5377970 0.91 BACE1 (0.66) BACE1CTSDCTSBBACE2
Hydrochloric Acid SCHEMBL5377965 0.91 BACE1 (0.66) BACE1CTSDCTSBBACE2
SCHEMBL5382113 0.90 BACE1 (0.68) BACE1CTSDCTSBBACE2
SCHEMBL5382108 0.90 BACE1 (0.68) BACE1CTSDCTSBBACE2
SCHEMBL3353057 0.90 BACE1 (0.69) BACE1CTSDCTSBBACE2
SCHEMBL3353049 0.90 BACE1 (0.69) BACE1CTSDCTSBBACE2
SCHEMBL3351304 0.88 BACE1 (0.67) BACE1CTSDCTSBBACE2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7176242-B2 N,N′-substituted-1,3-diamino-2-hydroxypropane derivatives ELAN PHARMACEUTICALS, INC. (US) 2007-02-13 US claimed
EP-1453789-A2 N,N'-SUBSTITUTED-1,3-DIAMINO-2-HYDROXYPROPANE DERIVATIVES Elan Pharmaceuticals, Inc. (US) 2004-09-08 EP claimed
WO-2003040096-A2 N, N'-SUBSTITUTED-1,3-DIAMINO-2-HYDROXYPROPANE DERIVATIVES ELAN PHARMACEUTICALS, INC. (US) 2003-05-15 WO claimed