SCHEMBL5375172

SCHEMBL5375172

Cc1nnc(-c2ccc3[nH]nc(-c4ccc(F)cc4)c3c2)o1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAP2K4 P45985 8/20 0.45
MAPK1 P28482 6/20 0.45
MAPKAPK3 Q16644 6/20 0.45
MAPK6 Q16659 6/20 0.45
MAPKAPK2 P49137 5/20 0.45
MAPKAPK5 Q8IW41 3/20 0.45
GUSB P08236 1/20 0.43
NTRK1 P04629 2/20 0.43
CSNK1D P48730 1/20 0.43
NPC1 O15118 1/20 0.42
RAB9A P51151 1/20 0.42
MKNK1 Q9BUB5 1/20 0.42
TLR8 Q9NR97 1/20 0.42
TLR7 Q9NYK1 1/20 0.42
NOTUM Q6P988 1/20 0.41
MAPT P10636 1/20 0.41
PIM1 P11309 1/20 0.40
PIM3 Q86V86 1/20 0.40
PIM2 Q9P1W9 1/20 0.40
HTR7 P34969 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13049888 0.89 MAP2K4 (0.54) MAP2K4MAPK1MAPKAPK3MAPK6MAPKAPK2
SCHEMBL5381615 0.84 MKNK1 (0.55) MAP2K4GUSBCSNK1DNPC1RAB9A
SCHEMBL25195476 0.82 TLR8 (0.46) MAP2K4MAPK1MAPKAPK3MAPK6MAPKAPK2
SCHEMBL5384307 0.78 CYP2C19 (0.48) MAP2K4CSNK1DTLR8TLR7PIM1
SCHEMBL5374591 0.77 MAP2K4 (0.71) MAP2K4MAPK1MAPKAPK3MAPK6MAPKAPK2
SCHEMBL2360473 0.76 NPC1 (0.72) GUSBNPC1RAB9ANOTUM
SCHEMBL16025795 0.75 LRRK2 (0.52)
SCHEMBL5372431 0.75 MAP2K4 (0.46) MAP2K4MAPK1MAPKAPK3MAPK6MAPKAPK2
SCHEMBL5390983 0.74 CSNK1D (0.52) CSNK1DTLR8TLR7MAPT
SCHEMBL23416052 0.74 MAPK14 (0.49) GUSBNPC1RAB9ANOTUMMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 39 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7211594-B2 Indazole compounds and compositions thereof as JNK inhibitors and for the treatment of diseases associated therewith SIGNAL PHARMACEUTICALS, LLC (US) 2007-05-01 US claimed
EP-1618093-A2 INDAZOLE DERIVATIVES AS JNK INHIBITORS Signal Pharmaceuticals LLC (US) 2006-01-25 EP claimed
WO-2004094388-A2 INDAZOLE DERIVATIVES AS JNK INHIBITORS SIGNAL PHARMACEUTICALS, LLC (US) 2004-11-04 WO claimed
US-20040127536-A1 Methods for treating an inflammatory condition or inhibiting JNK SIGNAL PHARMACEUTICALS, LLC 2004-07-01 US claimed
US-20170327788-A1 COMPOSITION FOR COLLECTING AND PRESERVING PLACENTAL STEM CELLS AND METHODS OF USING THE COMPOSITION ANTHROGENESIS CORPORATION (US) 2017-11-16 US disclosed
US-9725694-B2 Composition for collecting and preserving placental stem cells and methods of using the composition ANTHROGENESIS CORPORATION (US) 2017-08-08 US disclosed
US-9598669-B2 Composition for collecting placental stem cells and methods of using the composition ANTHROGENESIS CORPORATION (US) 2017-03-21 US disclosed
WO-2008091925-A2 TREATMENT OF AORTIC DISSECTION OR ANEURYSM COOK INCORPORATED (US) 2008-07-31 WO disclosed
WO-2007079185-A2 IMPROVED COMPOSITION FOR COLLECTING AND PRESERVING PLACENTAL STEM CELLS AND METHODS OF USING THE COMPOSITION ANTHROGENESIS CORPORATION (US) 2007-07-12 WO disclosed
US-7220771-B2 Methods of using indazole derivatives as JNK inhibitors SIGNAL PHARMACEUTICALS, LLC (US) 2007-05-22 US disclosed
US-7220771-B2 Methods of using indazole derivatives as JNK inhibitors SIGNAL PHARMACEUTICALS, LLC (US) 2007-05-22 US disclosed
US-7220771-B2 Methods of using indazole derivatives as JNK inhibitors SIGNAL PHARMACEUTICALS, LLC (US) 2007-05-22 US disclosed
WO-2004041191-A2 METHODS FOR THE TREATMENT, PREVENTION AND MANAGEMENT OF MACULAR DEGENERATION CELGENE CORPORATION (US) 2004-05-21 WO disclosed
US-20040087642-A1 Methods of using and compositions comprising a JNK inhibitor for the treatment, prevention, management and/or modification of pain CELGENE CORPORATION 2004-05-06 US disclosed
US-20040087642-A1 Methods of using and compositions comprising a JNK inhibitor for the treatment, prevention, management and/or modification of pain CELGENE CORPORATION 2004-05-06 US disclosed
US-20040077877-A1 Indazole derivatives as JNK inhibitors and compositions and methods related thereto SIGNAL PHARMACEUTICALS, INC. 2004-04-22 US disclosed
WO-2003102151-A2 MODULATING CELL DIFFERENTIATION AND TREATING MYELOPROLIFERTIVE DISORDERS WITH JNK/MKK INHIBITORS CELGENE CORPORATION (US) 2003-12-11 WO disclosed
WO-2003099221-A2 METHODS FOR USING JNK INHIBITORS FOR TREATING OR PREVENTING DISEASE-RELATED WASTING SIGNAL PHARMACEUTICALS, INC. (US) 2003-12-04 WO disclosed
WO-2002010137-A9 INDAZOLE DERIVATIVES AS JNK INHIBITORS SIGNAL PHARM INC (US) 2003-02-06 WO disclosed
US-20020103229-A1 Indazole derivatives as JNK inhibitors and compositions and methods related thereto SIGNAL PHARMACEUTICALS, LLC 2002-08-01 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040127536-A1 Methods for treating an inflammatory condition or inhibiting JNK MAPK1, MAP3K1, MAPKAPK2 MAP2K4 130/4885MAPK1 1/4885MAPKAPK3 13/4885
US-20040077877-A1 Indazole derivatives as JNK inhibitors and compositions and methods related thereto MAP3K7, MAP3K1, MAP3K8 MAP2K4 71/4885MAPK1 16/4885MAPKAPK3 21/4885
US-20040087642-A1 Methods of using and compositions comprising a JNK inhibitor for the treatment, prevention, management and/or modification of pain MAP3K1, MAP3K6, MAPKAPK2 MAP2K4 50/4885MAPK1 26/4885MAPKAPK3 21/4885
US-20020103229-A1 Indazole derivatives as JNK inhibitors and compositions and methods related thereto MAP3K7, MAP3K1, MAP3K8 MAP2K4 71/4885MAPK1 16/4885MAPKAPK3 21/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.