SCHEMBL5402043

SCHEMBL5402043

Cn1nc(-c2ccccc2)c2cccc(C(F)(F)F)c21

nearest known ligand 0.54

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 5/20 0.54
NR1H2 P55055 1/20 0.47
NR1H3 Q13133 1/20 0.47
ALDH1A1 P00352 3/20 0.45
KDM4E B2RXH2 2/20 0.45
HSD11B1 P28845 1/20 0.43
LMNA P02545 1/20 0.42
NPSR1 Q6W5P4 1/20 0.42
RORC P51449 3/20 0.41
SSTR4 P31391 1/20 0.41
ADORA3 P0DMS8 2/20 0.41
ADORA1 P30542 2/20 0.41
POLB P06746 1/20 0.41
HPGD P15428 1/20 0.40
PPARG P37231 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4028983 0.88 ESR1 (0.70) ESR1RORCSSTR4HPGDPPARG
SCHEMBL4027587 0.82 ESR1 (0.53) ESR1NR1H2NR1H3ALDH1A1LMNA
SCHEMBL13106136 0.79 SSTR4 (0.44) ESR1NR1H2NR1H3HSD11B1SSTR4
SCHEMBL13202563 0.79 SSTR4 (0.44) ESR1NR1H2NR1H3ALDH1A1HSD11B1
SCHEMBL4027869 0.76 ESR1 (0.65) ESR1SSTR4SMN1; SMN2
SCHEMBL29941523 0.75 ESR1 (0.66) ESR1NR1H2NR1H3ALDH1A1LMNA
SCHEMBL21067954 0.75 ESR1 (0.66) ESR1NR1H2NR1H3ALDH1A1LMNA
SCHEMBL16252840 0.74 SSTR4 (0.41) ESR1NR1H2NR1H3ALDH1A1HSD11B1
SCHEMBL16252859 0.74 SSTR4 (0.51) ESR1NR1H2NR1H3HSD11B1SSTR4
SCHEMBL15631890 0.73 KMT2A (0.65) ESR1NR1H2NR1H3ALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7241791-B2 Substituted 4-(indazol-3-yl)phenols WYETH (US) 2007-07-10 US disclosed