SCHEMBL5406598

SCHEMBL5406598

O=C(NS(=O)(=O)/C=C/c1ccc(Cl)cc1)c1ccc(F)cc1C(F)(F)F

nearest known ligand 0.51

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
FLT1 P17948 5/20 0.51
FLT4 P35916 5/20 0.51
KDR P35968 5/20 0.51
PTGES2 Q9H7Z7 8/20 0.47
MAOB P27338 1/20 0.44
KCNA3 P22001 2/20 0.38
DRD2 P14416 1/20 0.37
DRD1 P21728 1/20 0.37
CYP3A4 P08684 1/20 0.37
NPC1 O15118 1/20 0.36
RAB9A P51151 1/20 0.36
MET P08581 1/20 0.36
PTGS2 P35354 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5406605 1.00 FLT1 (0.51) FLT1FLT4KDRPTGES2MAOB
SCHEMBL5418917 0.90 PTGES2 (0.52) FLT1FLT4KDRPTGES2MAOB
SCHEMBL5418925 0.90 PTGES2 (0.52) FLT1FLT4KDRPTGES2MAOB
SCHEMBL5403851 0.89 FLT1 (0.66) FLT1FLT4KDRPTGES2RAB9A
SCHEMBL4620014 0.88 KMT2A (0.47) FLT1FLT4KDRPTGES2MAOB
SCHEMBL4620007 0.88 KMT2A (0.47) FLT1FLT4KDRPTGES2MAOB
SCHEMBL5408883 0.88 PTGES2 (0.50) FLT1FLT4KDRPTGES2DRD2
SCHEMBL5408893 0.88 PTGES2 (0.50) FLT1FLT4KDRPTGES2DRD2
SCHEMBL5411552 0.86 FLT1 (0.53) FLT1FLT4KDRPTGES2MAOB
SCHEMBL5411563 0.86 FLT1 (0.53) FLT1FLT4KDRPTGES2MAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7208526-B2 For example, (E)-2-(4-Chloro-phenyl)-ethenesulfonic acid 2,4-dichloro-benzoylamide; for use in the control or prevention of illnesses such as cancer; antitumor agents HOFFMANN-LA ROCHE INC. (US) 2007-04-24 US claimed
US-20060270874-A1 Styrylsulfonamides HOFFMANN-LA ROCHE INC. 2006-11-30 US claimed
US-7208526-B2 For example, (E)-2-(4-Chloro-phenyl)-ethenesulfonic acid 2,4-dichloro-benzoylamide; for use in the control or prevention of illnesses such as cancer; antitumor agents HOFFMANN-LA ROCHE INC. (US) 2007-04-24 US disclosed
US-20060270874-A1 Styrylsulfonamides HOFFMANN-LA ROCHE INC. 2006-11-30 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060270874-A1 Styrylsulfonamides STS, SULT1E1, BRCA1 FLT1 4126/4885FLT4 4438/4885KDR 4332/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.