SCHEMBL545938

SCHEMBL545938

CC1=C[N]C(=S)NC1=O

nearest known ligand 0.00

⚠ Novel chemotype — no close known analogue (best Tanimoto < 0.3). Unexplored chemical space relative to ChEMBL.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6513508 0.70
SCHEMBL545940 0.68
SCHEMBL7699279 0.57
SCHEMBL36967 0.57
SCHEMBL996566 0.57 GSK3A (0.33)
SCHEMBL3541281 0.55 GSK3B (0.48)
SCHEMBL2042092 0.55
Ethane SCHEMBL21589349 0.55 GSK3A (0.32)
SCHEMBL13970731 0.52
SCHEMBL12472456 0.52

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 135 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20070179100-A1 Protected monomers ALNYLAM PHARMACEUTICALS, INC. 2007-08-02 US claimed
EP-1625138-A2 PROTECTED MONOMERS Alnylam Pharmaceuticals Inc. (US) 2006-02-15 EP claimed
EP-1499627-A2 NUCLEASE RESISTANT CHIMERIC OLIGONUCLEOTIDES ISIS Pharmaceuticals, Inc. (US) 2005-01-26 EP claimed
WO-2004094345-A2 PROTECTED MONOMERS ALNYLAM PHARMACEUTICALS INC. (US) 2004-11-04 WO claimed
US-20040033973-A1 Compounds and oligomeric compounds comprising novel nucleobases ISIS PHARMACEUTICALS, INC. 2004-02-19 US claimed
US-20030207804-A1 Modified peptide nucleic acids ISIS PHARMACEUTICALS, INC. 2003-11-06 US claimed
US-20030175906-A1 Nuclease resistant chimeric oligonucleotides ISIS PHARMACEUTICALS, INC. 2003-09-18 US claimed
US-20030158403-A1 Nuclease resistant chimeric oligonucleotides ISIS PHARMACEUTICALS, INC. 2003-08-21 US claimed
WO-2003004602-A2 NUCLEASE RESISTANT CHIMERIC OLIGONUCLEOTIDES ISIS PHARMACEUTICALS, INC. (US) 2003-01-16 WO claimed
WO-2002097134-A2 MODIFIED PEPTIDE NUCLEIC ACID ISIS PHARMACEUTICALS, INC. (US) 2002-12-05 WO claimed
WO-2024135721-A1 METHOD FOR PRODUCING PRODUCTION INTERMEDIATE, PRODUCTION INTERMEDIATE THEREOF, AND METHOD FOR PRODUCING CROSSLINKED ARTIFICIAL NUCLEIC ACID INTERMEDIATE BY USING SAME 田辺三菱製薬株式会社 2024-06-27 WO disclosed
US-11814407-B2 Multiple coupling and oxidation method ROCHE INNOVATION CENTER COPENHAGEN A/S (CH) 2023-11-14 US disclosed
US-20220403377-A1 MODIFIED iRNA AGENTS ALNYLAM PHARMACEUTICALS, INC. 2022-12-22 US disclosed
US-11530408-B2 Therapeutic compositions ALNYLAM PHARMACEUTICALS, INC. (US) 2022-12-20 US disclosed
US-11312957-B2 Modified iRNA agents ALNYLAM PHARMACEUTICALS, INC. (US) 2022-04-26 US disclosed
WO-2004090108-A2 IRNA CONJUGATES ALNYLAM PHARMACEUTICALS (US) 2004-10-21 WO disclosed
WO-2004080406-A2 THERAPEUTIC COMPOSITIONS ALNYLAM PHARMACEUTICALS (US) 2004-09-23 WO disclosed
US-20040033973-A1 Compounds and oligomeric compounds comprising novel nucleobases ISIS PHARMACEUTICALS, INC. 2004-02-19 US disclosed
US-20030207804-A1 Modified peptide nucleic acids ISIS PHARMACEUTICALS, INC. 2003-11-06 US disclosed
WO-2002097134-A2 MODIFIED PEPTIDE NUCLEIC ACID ISIS PHARMACEUTICALS, INC. (US) 2002-12-05 WO disclosed