SCHEMBL5472811

SCHEMBL5472811

O=C1Nc2ccc(Cl)cc2C1=Cc1ccc(Cl)cc1Cl

nearest known ligand 0.65

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
LRRK2 Q5S007 6/20 0.65
MDM2 Q00987 5/20 0.63
PSEN1 P49768 2/20 0.62
PSEN2 P49810 2/20 0.62
APH1B Q8WW43 2/20 0.62
NCSTN Q92542 2/20 0.62
APH1A Q96BI3 2/20 0.62
PSENEN Q9NZ42 2/20 0.62
PDGFRB P09619 1/20 0.60
RPS6KA3 P51812 1/20 0.59
RET P07949 1/20 0.58
IDO1 P14902 1/20 0.57
TDO2 P48775 1/20 0.57
TGM2 P21980 1/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5472809 1.00 LRRK2 (0.65) LRRK2MDM2PSEN1PSEN2APH1B
SCHEMBL7138970 0.90 LRRK2 (0.54) LRRK2MDM2PSEN1PSEN2APH1B
SCHEMBL14448904 0.88 FLT3 (0.59) LRRK2MDM2PDGFRBRPS6KA3RET
SCHEMBL5472208 0.88 FLT3 (0.59) LRRK2MDM2PDGFRBRPS6KA3RET
SCHEMBL5472209 0.88 FLT3 (0.59) LRRK2MDM2PDGFRBRPS6KA3RET
SCHEMBL5469641 0.88 LRRK2 (0.70) LRRK2MDM2PSEN1PSEN2APH1B
SCHEMBL5469637 0.88 LRRK2 (0.70) LRRK2MDM2PSEN1PSEN2APH1B
SCHEMBL7135626 0.86 MDM2 (0.50) LRRK2MDM2PSEN1PSEN2APH1B
SCHEMBL7139608 0.83 SRC (0.54) LRRK2MDM2PDGFRBRPS6KA3RET
SCHEMBL5477805 0.81 LRRK2 (0.83) LRRK2PSEN1PSEN2APH1BNCSTN

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20070167488-A1 Novel therapeutic use LEO PHARMA A/S (DK) 2007-07-19 US claimed
EP-1696906-A1 NOVEL THERAPEUTIC USE OF INDOLINONE DERIVATIVES Leo Pharma A/S (DK) 2006-09-06 EP claimed
WO-2005058309-A1 NOVEL THERAPEUTIC USE OF INDOLINONE DERIVATIVES LEO PHARMA A/S (DK) 2005-06-30 WO claimed
US-20070167488-A1 Novel therapeutic use LEO PHARMA A/S (DK) 2007-07-19 US disclosed
EP-1696906-A1 NOVEL THERAPEUTIC USE OF INDOLINONE DERIVATIVES Leo Pharma A/S (DK) 2006-09-06 EP disclosed
WO-2005058309-A1 NOVEL THERAPEUTIC USE OF INDOLINONE DERIVATIVES LEO PHARMA A/S (DK) 2005-06-30 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070167488-A1 Novel therapeutic use MAG, PMP22, MYT1 LRRK2 1753/4885MDM2 4274/4885PSEN1 1618/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.