SCHEMBL5480090

SCHEMBL5480090

Cc1c(Cl)ccc2c1NC(=S)C2(c1ccc(N(C)C)cc1)c1ccc(N(C)C)cc1

nearest known ligand 0.32

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HTR6 P50406 1/20 0.32
CES1 P23141 1/20 0.32
FLI1 Q01543 1/20 0.31
EWSR1 Q01844 1/20 0.31
ALDH1A1 P00352 3/20 0.31
TSHR P16473 2/20 0.31
HSD17B10 Q99714 2/20 0.31
CYP3A4 P08684 1/20 0.31
HPGD P15428 1/20 0.31
HIF1A Q16665 1/20 0.31
TDP1 Q9NUW8 1/20 0.31
ALOX15 P16050 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5482232 0.83 MAPT (0.33) CES1ALDH1A1
SCHEMBL5477636 0.83 CNR1 (0.40) CES1
SCHEMBL5480076 0.76 MAPT (0.43) CES1ALDH1A1HSD17B10CYP3A4
SCHEMBL5482277 0.76 SMN1; SMN2 (0.43) ALDH1A1TSHRCYP3A4TDP1
SCHEMBL5479391 0.76 CES1 (0.34) CES1HPGD
SCHEMBL5478235 0.68 HTT (0.46) CES1ALDH1A1TSHRALOX15
SCHEMBL5475160 0.66 POLB (0.44) CES1ALDH1A1TSHRALOX15
SCHEMBL5475401 0.66 HTT (0.43) CES1ALDH1A1TSHRALOX15
SCHEMBL5474643 0.66 CNR1 (0.61) HTR6CES1ALDH1A1TSHRALOX15
SCHEMBL5474437 0.63 CNR1 (0.57) HTR6CES1ALDH1A1TSHRALOX15

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20070299102-A1 Diphenyl Ox-Indol-2-One Compounds and Their Use in the Treatment of Cancer TOPO TARGET A/S (DK) 2007-12-27 US claimed
US-20070299102-A1 Diphenyl Ox-Indol-2-One Compounds and Their Use in the Treatment of Cancer TOPO TARGET A/S (DK) 2007-12-27 US disclosed
EP-1734951-A2 DIPHENYL-INDOL-2-ON COMPOUNDS AND THEIR USE IN THE TREATMENT OF CANCER TopoTarget A/S (DK) 2006-12-27 EP disclosed
WO-2005097107-A2 DIPHENYL - INDOL-2-ON COMPOUNDS AND THEIR USE IN THE TREATMENT OF CANCER TOPOTARGET A/S (DK) 2005-10-20 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070299102-A1 Diphenyl Ox-Indol-2-One Compounds and Their Use in the Treatment of Cancer MTOR, RICTOR, CDK4 HTR6 639/4885CES1 4132/4885FLI1 538/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.