SCHEMBL5484694

SCHEMBL5484694

O=c1ccc([C@H]2O[C@H](CO)[C@@H](O)[C@H]2O)c[nH]1

nearest known ligand 0.50

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
SLC5A2 P31639 19/20 0.50
SLC28A1 O00337 1/20 0.42
SLC28A2 O43868 1/20 0.42
SLC29A1 Q99808 1/20 0.42
SLC28A3 Q9HAS3 1/20 0.42
SLC5A1 P13866 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16781781 1.00 SLC5A2 (0.50) SLC5A2SLC28A1SLC28A2SLC29A1SLC28A3
SCHEMBL18870681 1.00 SLC5A2 (0.50) SLC5A2SLC28A1SLC28A2SLC29A1SLC28A3
SCHEMBL16631540 1.00 SLC5A2 (0.50) SLC5A2SLC28A1SLC28A2SLC29A1SLC28A3
SCHEMBL5487423 1.00 SLC5A2 (0.50) SLC5A2SLC28A1SLC28A2SLC29A1SLC28A3
SCHEMBL17082382 1.00 SLC5A2 (0.50) SLC5A2SLC28A1SLC28A2SLC29A1SLC28A3
SCHEMBL16631946 1.00 SLC5A2 (0.50) SLC5A2SLC28A1SLC28A2SLC29A1SLC28A3
SCHEMBL16631566 0.87 CDA (0.40) SLC5A2SLC28A1SLC28A2SLC29A1SLC28A3
SCHEMBL18079914 0.84 SLC5A2 (0.44) SLC5A2SLC5A1
SCHEMBL18870679 0.81 SLC5A2 (0.35) SLC5A2
SCHEMBL17378615 0.81 SLC5A2 (0.35) SLC5A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-3903392-B2 2007-04-11 JP claimed
US-6248878-B1 INCLUDING BASES 2-FLUOROPYRIDINE-3-YL, PYRIDINE-2-ONE-3-YL, PYRIDIN-2-(4-NITROPHENYLETHYL)-ONE-3-YL, 2-BROMOPYRIDINE-5-YL , PYRIDIN-2-ONE-5-YL, 2-AMINOPYRIDINE-5-YL, PYRIDIN-2-(4-NITROPHENYLETHYL)-ONE-5-YL; ANTISENSE/ANTICANCER AGENTS RIBOZYME PHARMACEUTICALS, INC. 2001-06-19 US claimed
JP-2001507688-A 2001-06-12 JP claimed
EP-0948511-A2 CHEMICAL SYNTHESIS OF NUCLEOSIDES ANALOGS AND THEIR INCORPORATION INTO POLYNUCLEOTIDES RIBOZYME PHARMACEUTICALS, INC. (US) 1999-10-13 EP claimed
WO-1998028317-A2 SYNTHESIS OF NUCLEOSIDES AND POLYNUCLEOTIDES RIBOZYME PHARMACEUTICALS, INC. (US) 1998-07-02 WO claimed
EP-0948511-B1 CHEMICAL SYNTHESIS OF NUCLEOSIDES ANALOGS AND THEIR INCORPORATION INTO POLYNUCLEOTIDES SIRNA THERAPEUTICS INC (US) 2006-10-18 EP disclosed
US-6248878-B1 INCLUDING BASES 2-FLUOROPYRIDINE-3-YL, PYRIDINE-2-ONE-3-YL, PYRIDIN-2-(4-NITROPHENYLETHYL)-ONE-3-YL, 2-BROMOPYRIDINE-5-YL , PYRIDIN-2-ONE-5-YL, 2-AMINOPYRIDINE-5-YL, PYRIDIN-2-(4-NITROPHENYLETHYL)-ONE-5-YL; ANTISENSE/ANTICANCER AGENTS RIBOZYME PHARMACEUTICALS, INC. 2001-06-19 US disclosed
US-6248878-B1 INCLUDING BASES 2-FLUOROPYRIDINE-3-YL, PYRIDINE-2-ONE-3-YL, PYRIDIN-2-(4-NITROPHENYLETHYL)-ONE-3-YL, 2-BROMOPYRIDINE-5-YL , PYRIDIN-2-ONE-5-YL, 2-AMINOPYRIDINE-5-YL, PYRIDIN-2-(4-NITROPHENYLETHYL)-ONE-5-YL; ANTISENSE/ANTICANCER AGENTS RIBOZYME PHARMACEUTICALS, INC. 2001-06-19 US disclosed
EP-0948511-A2 CHEMICAL SYNTHESIS OF NUCLEOSIDES ANALOGS AND THEIR INCORPORATION INTO POLYNUCLEOTIDES RIBOZYME PHARMACEUTICALS, INC. (US) 1999-10-13 EP disclosed
WO-1998028317-A2 SYNTHESIS OF NUCLEOSIDES AND POLYNUCLEOTIDES RIBOZYME PHARMACEUTICALS, INC. (US) 1998-07-02 WO disclosed