SCHEMBL5488267

SCHEMBL5488267

NCC1(Cc2ccc3[nH]c(-c4n[nH]c5cc(-c6nnn[nH]6)ccc45)cc3c2)CCNCC1

nearest known ligand 0.44

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
CHEK1 O14757 20/20 0.44
CDK7 P50613 15/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5054048 0.81 CHEK1 (0.62) CHEK1CDK7
SCHEMBL5054012 0.76 CHEK1 (0.69) CHEK1CDK7
SCHEMBL144041 0.74 CHEK1 (0.68) CHEK1CDK7
SCHEMBL4156767 0.73 CHEK1 (0.58) CHEK1CDK7
SCHEMBL4159485 0.73 CHEK1 (0.77) CHEK1CDK7
SCHEMBL5055589 0.72 CHEK1 (0.64) CHEK1CDK7
SCHEMBL5054083 0.72 CHEK1 (0.57) CHEK1CDK7
SCHEMBL4125079 0.63 ITK (0.68) CHEK1CDK7
SCHEMBL5061267 0.62 CHEK1 (0.78) CHEK1CDK7
SCHEMBL5058797 0.62 CHEK1 (0.76) CHEK1CDK7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1851203-A2 INHIBITORS OF CHECKPOINT KINASES Merck & Co., Inc. (US) 2007-11-07 EP disclosed
WO-2006086255-A2 INHIBITORS OF CHECKPOINT KINASES MERCK & CO., INC. (US) 2006-08-17 WO disclosed