SCHEMBL5489529

SCHEMBL5489529

CSc1nc2ccc(S(=O)(=O)NCl)cc2o1

nearest known ligand 0.51

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.36
ELANE P08246 2/20 0.36
LMNA P02545 5/20 0.35
MAPT P10636 4/20 0.35
TP53 P04637 3/20 0.35
POLB P06746 2/20 0.35
KMT2A Q03164 1/20 0.35
FBP1 P09467 3/20 0.35
HTT P42858 3/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
HSP90AA1 P07900 1/20 0.34
HPGD P15428 1/20 0.34
TSHR P16473 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14508206 0.84 ELANE (0.39) ALDH1A1ELANELMNAMAPTTP53
SCHEMBL14508173 0.82 ELANE (0.40) ALDH1A1ELANELMNAMAPTKMT2A
SCHEMBL14608770 0.78 KMT2A (0.38) ALDH1A1ELANELMNAPOLBKMT2A
SCHEMBL14608741 0.73 HTT (0.41) ALDH1A1LMNAPOLBHTTSMN1; SMN2
SCHEMBL12384123 0.72 PIK3CG (0.56) ELANELMNAMAPTTP53POLB
SCHEMBL1748063 0.71 KDM4E (0.56) ALDH1A1ELANEMAPTTP53KMT2A
SCHEMBL4704291 0.70 MAPT (0.56) ALDH1A1LMNAMAPTKMT2AHTT
SCHEMBL3573726 0.70 HTT (0.50) ALDH1A1LMNAPOLBKMT2AHTT
SCHEMBL14985575 0.70 HTT (0.50) ALDH1A1LMNAMAPTPOLBKMT2A
SCHEMBL1563928 0.69 ESR1 (0.53)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1858901-A1 BENZOTHIAZOLE, THIAZOLOPYRIDINE, BENZOOXAZOLE AND OXAZOLOPYRIDINE DERIVATIVES AS ANTIDIABETIC COMPOUNDS F. Hoffmann-La Roche AG (CH) 2007-11-28 EP disclosed
WO-2006094682-A1 BENZOTHIAZOLE, THIAZOLOPYRIDINE, BENZOOXAZOLE AND OXAZOLOPYRIDINE DERIVATIVES AS ANTIDIABETIC COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2006-09-14 WO disclosed