SCHEMBL5491699

SCHEMBL5491699

CCOC(=O)C(=CNc1cc(OC)ccc1Br)C(=O)OCC.CCOC(=O)c1c[nH]c2c(Br)ccc(OC)c2c1=O

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.48
GAA P10253 3/20 0.48
ALDH1A1 P00352 3/20 0.48
HPGD P15428 2/20 0.48
NPSR1 Q6W5P4 1/20 0.47
LMNA P02545 3/20 0.46
MAPT P10636 3/20 0.46
THRB P10828 2/20 0.40
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40
GABRA1 P14867 1/20 0.39
GABRB1 P18505 1/20 0.39
GABRA3 P34903 1/20 0.39
GABRB2 P47870 1/20 0.39
CLEC4M Q9H2X3 1/20 0.38
DHODH Q02127 1/20 0.38
CYP3A4 P08684 2/20 0.38
CYP1A2 P05177 1/20 0.38
CYP2C19 P33261 1/20 0.38
JAK3 P52333 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL397393 0.83 CLEC4M (0.52) KDM4EALDH1A1HPGDMAPTMEN1
SCHEMBL396592 0.81 KDM4E (0.66) KDM4EGAAALDH1A1HPGDNPSR1
SCHEMBL10862234 0.77 KDM4E (0.76) KDM4EGAAALDH1A1HPGDNPSR1
SCHEMBL9829849 0.75 CLEC4M (0.56) KDM4EALDH1A1HPGDMAPTMEN1
SCHEMBL2035901 0.72 CLEC4M (0.55) KDM4EALDH1A1HPGDMAPTMEN1
SCHEMBL10860624 0.70 MEN1 (0.60) KDM4EGAAALDH1A1NPSR1LMNA
SCHEMBL2488117 0.70 CLEC4M (0.53) KDM4EALDH1A1HPGDMAPTMEN1
SCHEMBL7291074 0.69 CLEC4M (0.50) KDM4EGAALMNAMAPTMEN1
SCHEMBL2970561 0.69 MEN1 (0.75) KDM4EGAAALDH1A1NPSR1LMNA
SCHEMBL62162 0.69 CLEC4M (0.52) KDM4EALDH1A1HPGDMAPTMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1773816-A2 MODULATORS OF ATP-BINDING CASSETTE TRANSPORTERS Vertex Pharmaceuticals Incorporated (US) 2007-04-18 EP disclosed
WO-2006002421-A2 MODULATORS OF ATP-BINDING CASSETTE TRANSPORTERS VERTEX PHARMACEUTICALS INCORPORATED (US) 2006-01-05 WO disclosed