SCHEMBL5493046

SCHEMBL5493046

COCCN(CCCOc1cc2ncnc(Nc3ccn(CC(=O)Nc4cccc(F)c4F)n3)c2cc1OC)CCOP(=O)(O)O

nearest known ligand 0.59

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
AURKA O14965 13/20 0.59
AURKB Q96GD4 4/20 0.59
HDAC3 O15379 4/20 0.48
KDR P35968 4/20 0.48
HDAC4 P56524 4/20 0.48
HDAC1 Q13547 4/20 0.48
HDAC7 Q8WUI4 4/20 0.48
HDAC2 Q92769 4/20 0.48
HDAC10 Q969S8 4/20 0.48
HDAC11 Q96DB2 4/20 0.48
HDAC8 Q9BY41 4/20 0.48
HDAC6 Q9UBN7 4/20 0.48
HDAC9 Q9UKV0 4/20 0.48
HDAC5 Q9UQL6 4/20 0.48
EGFR P00533 2/20 0.48
MAPK14 Q16539 1/20 0.45
ERBB2 P04626 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2053398 0.89 AURKA (0.61) AURKAAURKBHDAC3KDRHDAC4
SCHEMBL3425998 0.89 AURKA (0.59) AURKAAURKBKDREGFR
SCHEMBL5039274 0.89 AURKA (0.74) AURKAAURKBHDAC3KDRHDAC4
SCHEMBL5043941 0.87 AURKA (0.59) AURKAAURKBHDAC3KDRHDAC4
SCHEMBL2048922 0.86 AURKA (0.62) AURKAAURKBHDAC3KDRHDAC4
SCHEMBL3489745 0.86 AURKA (0.80) AURKAAURKBKDREGFR
Hydrochloric Acid SCHEMBL5048426 0.86 AURKA (0.58) AURKAAURKBHDAC3KDRHDAC4
SCHEMBL5491653 0.85 AURKA (0.62) AURKAAURKBKDREGFRERBB2
SCHEMBL6020449 0.85 AURKA (0.62) AURKAAURKBHDAC3KDRHDAC4
SCHEMBL2050510 0.85 AURKA (0.67) AURKAAURKBKDREGFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1578755-B1 PHOSPHONOOXY QUINAZOLINE DERIVATIVES AND THEIR PHARMACEUTICAL USE ASTRAZENECA AB (SE) 2007-08-22 EP disclosed