SCHEMBL5494359

SCHEMBL5494359

CC(C)Oc1cc(C(F)(F)F)c2c3c(ccc2n1)NC(C(C)C)CO3

nearest known ligand 0.40

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
AR P10275 10/20 0.40
CDK1 P06493 1/20 0.31
TRPA1 O75762 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5118678 1.00 AR (0.40) ARCDK1TRPA1
SCHEMBL5114827 0.89 AR (0.53) ARCDK1TRPA1
SCHEMBL5114835 0.89 AR (0.53) ARCDK1TRPA1
SCHEMBL5122002 0.86 AR (0.55) ARCDK1
SCHEMBL5124748 0.86 AR (0.55) ARCDK1
SCHEMBL5116557 0.85 AR (0.45) AR
SCHEMBL5123270 0.84 AR (0.56) AR
SCHEMBL5486825 0.84 AR (0.55) ARCDK1TRPA1
SCHEMBL5115984 0.84 AR (0.55) ARCDK1TRPA1
SCHEMBL5123257 0.82 AR (0.42) ARCDK1TRPA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7214690-B2 Tricyclic quinolinone and tricyclic quinoline androgen receptor modulator compounds and methods LIGAND PHARMACEUTICALS INCORPORATED (US) 2007-05-08 US disclosed