Oxybutynin

Oxybutynin

SCHEMBL5494388

CCN(CC)CC#CCOC(=O)C(O)(c1ccccc1)C1CCCCC1.CCN(CC)CC#CCOC(=O)C(O)(c1ccccc1)C1CCCCC1.Cl

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

CHRM2CHRM3

The experimentally established mechanism targets of Oxybutynin. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRM2 known ✓ P08172 6/20 0.98
CHRM3 known ✓ P20309 4/20 0.98
MEN1 O00255 1/20 1.00
RECQL P46063 1/20 1.00
PMP22 Q01453 1/20 1.00
KMT2A Q03164 1/20 1.00
NPSR1 Q6W5P4 1/20 1.00
CHRM1 P11229 6/20 0.98
CHRM4 P08173 4/20 0.98
KCNH2 Q12809 3/20 0.98
CYP2C19 P33261 2/20 0.98
SLC6A3 Q01959 2/20 0.98
CYP3A4 P08684 2/20 0.98
CYP1A2 P05177 1/20 0.98
CYP2D6 P10635 1/20 0.98
CYP2C9 P11712 1/20 0.98
PKM P14618 1/20 0.98
NFKB1 P19838 1/20 0.98
THPO P40225 1/20 0.98
ABCB11 O95342 1/20 0.98

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Esoxybutynin SCHEMBL5690091 1.00 MEN1 (1.00) MEN1RECQLPMP22KMT2ANPSR1
Aroxybutynin SCHEMBL27093068 1.00 MEN1 (1.00) MEN1RECQLPMP22KMT2ANPSR1
Oxybutynin SCHEMBL8019436 1.00 MEN1 (1.00) MEN1RECQLPMP22KMT2ANPSR1
Oxybutynin SCHEMBL25751 1.00 MEN1 (1.00) MEN1RECQLPMP22KMT2ANPSR1
Oxybutynin SCHEMBL1560964 0.99 CHRM2 (1.00) MEN1RECQLPMP22KMT2ANPSR1
Esoxybutynin SCHEMBL290373 0.99 CHRM2 (1.00) MEN1RECQLPMP22KMT2ANPSR1
Oxybutynin SCHEMBL2992 0.99 CHRM2 (1.00) MEN1RECQLPMP22KMT2ANPSR1
Aroxybutynin SCHEMBL25880 0.99 CHRM2 (1.00) MEN1RECQLPMP22KMT2ANPSR1
Oxybutynin SCHEMBL7557853 0.98 CHRM2 (0.98) MEN1RECQLPMP22KMT2ANPSR1
Oxybutynin SCHEMBL7895841 0.98 CHRM2 (0.98) MEN1RECQLPMP22KMT2ANPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1737539-A1 THERAPEUTIC COMBINATION FOR TREATMENT OF ALZHEIMERS DISEASE Warner-Lambert Company LLC (US) 2007-01-03 EP disclosed
WO-2005099823-A1 THERAPEUTIC COMBINATION FOR TREATMENT OF ALZHEIMERS DISEASE WARNER-LAMBERT COMPANY LLC (US) 2005-10-27 WO disclosed