SCHEMBL5497570

SCHEMBL5497570

CCCc1ccccc1Oc1ccc(C#N)cc1Cl.Cc1cc(C)c(Oc2ccc(C#N)cc2Cl)c(C)c1

nearest known ligand 0.59

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
AR P10275 4/20 0.59
SLC6A4 P31645 11/20 0.46
SLC6A3 Q01959 9/20 0.46
KCNH2 Q12809 2/20 0.46
SLC6A2 P23975 8/20 0.41
HTR2A P28223 1/20 0.38
TBXA2R P21731 1/20 0.38
CHRM1 P11229 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4163791 0.90 AR (0.64) ARSLC6A4SLC6A3KCNH2SLC6A2
SCHEMBL4179861 0.83 AR (0.64) ARSLC6A4SLC6A3KCNH2HTR2A
SCHEMBL4178705 0.80 AR (0.68) ARSLC6A4SLC6A3KCNH2SLC6A2
SCHEMBL4181001 0.76 AR (0.73) ARSLC6A4SLC6A3KCNH2HTR2A
SCHEMBL4168825 0.76 AR (1.00) ARSLC6A4SLC6A3KCNH2SLC6A2
SCHEMBL4181543 0.73 AR (0.73) ARSLC6A4SLC6A3KCNH2HTR2A
SCHEMBL4179847 0.72 AR (0.68) ARSLC6A4SLC6A3KCNH2SLC6A2
SCHEMBL5503503 0.72 AR (0.56) ARSLC6A4SLC6A3KCNH2SLC6A2
SCHEMBL25451306 0.71 AR (0.60) ARSLC6A4SLC6A3KCNH2SLC6A2
SCHEMBL18164415 0.71 SLC6A4 (0.49) ARSLC6A4SLC6A3SLC6A2HTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1781280-A2 ANDROGEN MODULATORS Warner-Lambert Company LLC (US) 2007-05-09 EP claimed
WO-2006018723-A2 ANDROGEN MODULATORS WARNER-LAMBERT COMPANY LLC (US) 2006-02-23 WO claimed