SCHEMBL5499353

SCHEMBL5499353

O=c1[nH]ccc2nc(-c3ccc(CN4CCC(c5c[nH]c(-c6ccccn6)n5)CC4)cc3)c(-c3ccccc3)cc12

nearest known ligand 0.74

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 5/20 0.74
AKT1 P31749 19/20 0.68
AKT2 P31751 12/20 0.68

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12759353 0.88 KCNH2 (0.72) KCNH2AKT1AKT2
SCHEMBL1059047 0.88 KCNH2 (0.76) KCNH2AKT1AKT2
Hydrochloric Acid SCHEMBL1501644 0.87 KCNH2 (0.75) KCNH2AKT1AKT2
SCHEMBL1501575 0.86 KCNH2 (0.72) KCNH2AKT1AKT2
SCHEMBL1501729 0.86 KCNH2 (0.71) KCNH2AKT1AKT2
SCHEMBL1501594 0.85 KCNH2 (0.77) KCNH2AKT1AKT2
SCHEMBL12759299 0.85 KCNH2 (0.72) KCNH2AKT1AKT2
SCHEMBL1501787 0.84 KCNH2 (0.71) KCNH2AKT1AKT2
SCHEMBL1501571 0.84 KCNH2 (0.71) KCNH2AKT1AKT2
SCHEMBL1501768 0.84 KCNH2 (0.68) KCNH2AKT1AKT2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1827436-A2 INHIBITORS OF AKT ACTIVITY Merck & Co., Inc. (US) 2007-09-05 EP disclosed
WO-2006065601-A2 INHIBITORS OF AKT ACTIVITY MERCK & CO., INC. (US) 2006-06-22 WO disclosed