SCHEMBL5500679

SCHEMBL5500679

COc1ccc(C(=O)C2CNc3ccccc32)cc1CSc1nc2cc(F)ccc2n1CC(=O)O

nearest known ligand 0.70

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
PTGDR2 Q9Y5Y4 20/20 0.70
CYP3A4 P08684 4/20 0.69
CYP2C9 P11712 3/20 0.63

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5113243 0.83 PTGDR2 (1.00) PTGDR2CYP3A4CYP2C9
SCHEMBL30538012 0.82 PTGDR2 (1.00) PTGDR2CYP3A4CYP2C9
SCHEMBL5122847 0.82 PTGDR2 (1.00) PTGDR2CYP3A4CYP2C9
SCHEMBL5121597 0.79 PTGDR2 (1.00) PTGDR2CYP3A4CYP2C9
SCHEMBL5106741 0.78 PTGDR2 (1.00) PTGDR2CYP3A4CYP2C9
SCHEMBL5110990 0.77 PTGDR2 (1.00) PTGDR2CYP3A4CYP2C9
SCHEMBL5121705 0.77 PTGDR2 (1.00) PTGDR2CYP3A4CYP2C9
SCHEMBL5120386 0.77 PTGDR2 (1.00) PTGDR2CYP3A4CYP2C9
SCHEMBL5113187 0.76 PTGDR2 (1.00) PTGDR2CYP3A4CYP2C9
SCHEMBL5114061 0.76 PTGDR2 (1.00) PTGDR2CYP3A4CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1784182-A1 2-SULFANYL-BENZIMIDAZOL-1-YL-ACETIC ACID DERIVATIVES AS CRTH2 ANTAGONISTS Actelion Pharmaceuticals Ltd. (CH) 2007-05-16 EP disclosed
WO-2006021418-A1 2-SULFANYL-BENZOIMIDAZOL-1-YL-ACETIC ACID DERIVATIVES AS CRTH2 ANTAGONISTS ACTELION PHARMACEUTICALS LTD (CH) 2006-03-02 WO disclosed