SCHEMBL5500905

SCHEMBL5500905

CCCC#Cc1cccc(OC(F)(F)F)c1

nearest known ligand 0.50

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 1/20 0.50
FFAR1 O14842 1/20 0.49
HAO1 Q9UJM8 3/20 0.46
ADORA2B P29275 3/20 0.41
CYP2D6 P10635 1/20 0.41
HRH3 Q9Y5N1 1/20 0.41
CTSS P25774 1/20 0.41
CTSK P43235 1/20 0.41
REN P00797 1/20 0.39
CTSD P07339 1/20 0.39
BACE1 P56817 1/20 0.39
BACE2 Q9Y5Z0 1/20 0.39
CHRM2 P08172 2/20 0.38
CHRM1 P11229 2/20 0.38
CHRM3 P20309 2/20 0.38
CETP P11597 3/20 0.37
GRM2 Q14416 1/20 0.36
CHRNB4 P30926 1/20 0.36
CHRNA3 P32297 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18834037 0.88 GRM5 (0.52) GRM5FFAR1HAO1ADORA2BCTSS
SCHEMBL3872159 0.82 FFAR1 (0.50) GRM5FFAR1HAO1BACE1CETP
SCHEMBL81119 0.81 FFAR1 (0.54) GRM5FFAR1HAO1ADORA2BCHRM2
SCHEMBL3874608 0.80 FFAR1 (0.67) GRM5FFAR1HAO1
SCHEMBL2232937 0.79 FFAR1 (0.56) GRM5FFAR1CHRM2CHRM1CHRM3
SCHEMBL16984726 0.79 GRM5 (0.56) GRM5FFAR1HAO1CTSSCTSK
SCHEMBL5481917 0.78 FFAR1 (0.44) GRM5FFAR1HAO1ADORA2BCHRM2
SCHEMBL13597746 0.76 GRM5 (0.53) GRM5FFAR1HAO1CYP2D6HRH3
SCHEMBL3937119 0.76 GRM5 (0.47) GRM5FFAR1ADORA2BCYP2D6HRH3
SCHEMBL4293314 0.75 GRM5 (0.48) GRM5FFAR1CHRM2CHRM1CHRM3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1765760-A1 PHENYL DERIVATIVES COMPRISING AN ACETYLENE GROUP F.HOFFMANN-LA ROCHE AG (CH) 2007-03-28 EP disclosed
WO-2006002802-A1 PHENYL DERIVATIVES COMPRISING AN ACETYLENE GROUP F. HOFFMANN-LA ROCHE AG (CH) 2006-01-12 WO disclosed