SCHEMBL5501902

SCHEMBL5501902

C=CCn1nc(-c2ccc(O)cc2O)c2cccc(C(F)(F)F)c21.C=CCn1nc(-c2ccc(OC)cc2OC)c2cccc(C(F)(F)F)c21

nearest known ligand 0.78

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 9/20 0.78
ESR2 Q92731 1/20 0.78
MAPT P10636 2/20 0.37
CNR1 P21554 1/20 0.37
CNR2 P34972 1/20 0.37
GPR55 Q9Y2T6 1/20 0.37
MEN1 O00255 2/20 0.35
KMT2A Q03164 2/20 0.35
MRGPRX4 Q96LA9 1/20 0.35
KDM4E B2RXH2 1/20 0.34
ALDH1A1 P00352 1/20 0.34
CYP3A4 P08684 1/20 0.34
HPGD P15428 1/20 0.34
HSD17B10 Q99714 1/20 0.34
CRHR1 P34998 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29817411 0.93 ESR1 (0.64) ESR1ESR2MAPTMEN1KMT2A
SCHEMBL3889569 0.93 ESR1 (0.64) ESR1ESR2MAPTMEN1KMT2A
SCHEMBL3890967 0.88 ESR1 (1.00) ESR1ESR2MAPTCNR1CNR2
SCHEMBL4030022 0.84 ESR1 (0.75) ESR1ESR2KDM4ECRHR1
SCHEMBL4032053 0.81 ESR1 (1.00) ESR1ESR2
SCHEMBL4029130 0.80 ESR1 (0.46) ESR1ESR2MAPTMEN1KMT2A
SCHEMBL4027158 0.79 ESR1 (0.45) ESR1ESR2MEN1KMT2AKDM4E
SCHEMBL4034557 0.79 ESR1 (0.44) ESR1ESR2MAPTMEN1KMT2A
SCHEMBL4031240 0.78 ESR1 (0.58) ESR1ESR2MAPTKDM4EALDH1A1
SCHEMBL4032697 0.77 ESR1 (0.43) ESR1ESR2CNR2MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1856151-A2 ESTROGEN RECEPTOR STRUCTURE Wyeth (US) 2007-11-21 EP disclosed
WO-2006078733-A2 ESTROGEN RECEPTOR STRUCTURE WYETH (US) 2006-07-27 WO disclosed