SCHEMBL5502415

SCHEMBL5502415

CC(=O)Nc1ccc(-c2nc(C(S)c3cccc(CCC(=O)NCCCN(C)C)n3)nc(N)c2C#N)cc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA1 P30542 2/20 0.47
ADORA2A P29274 2/20 0.47
ADORA3 P0DMS8 1/20 0.36
ADORA2B P29275 1/20 0.36
IKBKB O14920 4/20 0.36
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33
JAK2 O60674 1/20 0.33
MAP4K4 O95819 2/20 0.33
MAPK8 P45983 2/20 0.33
ITK Q08881 2/20 0.33
CLK4 Q9HAZ1 2/20 0.33
CHUK O15111 1/20 0.33
PRKD3 O94806 1/20 0.33
CDK2 P24941 1/20 0.33
MAPK9 P45984 1/20 0.33
CLK2 P49760 1/20 0.33
MAPK10 P53779 1/20 0.33
MAP4K2 Q12851 1/20 0.33
PASK Q96RG2 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL945978 0.96 ADORA1 (0.47) ADORA1ADORA2AADORA3ADORA2BIKBKB
Hydrochloric Acid SCHEMBL948352 0.95 ADORA1 (0.47) ADORA1ADORA2AADORA3ADORA2BIKBKB
SCHEMBL945760 0.90 ADORA1 (0.56) ADORA1ADORA2AADORA3ADORA2BIKBKB
Hydrochloric Acid SCHEMBL945957 0.90 ADORA1 (0.45) ADORA1ADORA2AADORA3ADORA2BIKBKB
SCHEMBL3737757 0.90 ADORA1 (0.45) ADORA1ADORA2AADORA3ADORA2BIKBKB
Hydrochloric Acid SCHEMBL946972 0.89 ADORA1 (0.55) ADORA1ADORA2AADORA3ADORA2BIKBKB
SCHEMBL946228 0.88 ADORA1 (0.45) ADORA1ADORA2AADORA3ADORA2BIKBKB
Hydrochloric Acid SCHEMBL946906 0.87 ADORA1 (0.45) ADORA1ADORA2AADORA3ADORA2BIKBKB
SCHEMBL950112 0.84 ADORA1 (0.46) ADORA1ADORA2AADORA3ADORA2BIKBKB
SCHEMBL3743152 0.83 ADORA1 (0.45) ADORA1ADORA2AADORA3ADORA2BIKBKB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1740574-B1 4-AMINO-5-CYANOPYRIMIDINE DERIVATIVES OTSUKA PHARMA CO LTD (JP) 2007-06-27 EP claimed