SCHEMBL5509150

SCHEMBL5509150

COc1cnc2cccc([C@@H](O)CN3CC4[C@@H](C3)[C@@H]4NCc3cc4ccccc4o3)c2n1

nearest known ligand 0.40

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 4/20 0.40
SLC2A1 P11166 4/20 0.36
DRD2 P14416 7/20 0.34
HTR2B P41595 7/20 0.34
HTR1A P08908 6/20 0.34
NPC1 O15118 1/20 0.33
RAB9A P51151 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5518086 0.81 KCNH2 (0.49) KCNH2SLC2A1
SCHEMBL5506820 0.76 KCNH2 (0.37) KCNH2SLC2A1
SCHEMBL3781930 0.73 SLC2A1 (0.52) KCNH2SLC2A1DRD2HTR2BHTR1A
SCHEMBL4495706 0.70 KCNH2 (0.47) KCNH2SLC2A1
SCHEMBL5516460 0.69 KCNH2 (0.61) KCNH2SLC2A1
SCHEMBL13921369 0.68 KCNH2 (0.81) KCNH2SLC2A1
SCHEMBL4489210 0.68 SLC2A1 (0.51) KCNH2SLC2A1
SCHEMBL5435565 0.68 KCNH2 (0.40) KCNH2SLC2A1
Hydrochloric Acid SCHEMBL6271264 0.68 KCNH2 (0.80) KCNH2SLC2A1
SCHEMBL5436003 0.67 KCNH2 (0.48) KCNH2SLC2A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1799676-A2 NEW BICYCLIC ANTIBIOTICS Actelion Pharmaceuticals Ltd. (CH) 2007-06-27 EP claimed
WO-2006032466-A2 NEW BICYCLIC ANTIBIOTICS ACTELION PHARMACEUTICALS LTD (CH) 2006-03-30 WO claimed