SCHEMBL5512650

SCHEMBL5512650

CC(C)c1nc(C(=O)C(=O)O)cs1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TLR7 Q9NYK1 1/20 0.50
HDAC1 Q13547 1/20 0.40
HDAC8 Q9BY41 1/20 0.40
HDAC6 Q9UBN7 1/20 0.40
PIK3CD O00329 1/20 0.38
PIK3CA P42336 1/20 0.38
PIK3CB P42338 1/20 0.38
PIK3CG P48736 1/20 0.38
KMT2A Q03164 2/20 0.38
GFER P55789 1/20 0.38
SLC6A3 Q01959 1/20 0.37
CHRM2 P08172 4/20 0.37
CHRM3 P20309 4/20 0.37
MEN1 O00255 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.35
L3MBTL1 Q9Y468 3/20 0.35
ALDH1A1 P00352 1/20 0.33
GAA P10253 1/20 0.32
MAPT P10636 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL314037 0.85 TLR7 (0.53) TLR7HDAC1HDAC8HDAC6PIK3CD
SCHEMBL5520327 0.84 TLR7 (0.49) TLR7HDAC1HDAC8HDAC6PIK3CD
SCHEMBL27830319 0.82 TLR7 (0.54) TLR7HDAC1HDAC8HDAC6PIK3CD
SCHEMBL13827949 0.81 TLR7 (0.53) TLR7HDAC1HDAC8HDAC6PIK3CD
SCHEMBL7029471 0.79 TLR7 (0.51) TLR7HDAC1HDAC8HDAC6PIK3CD
SCHEMBL21448923 0.79 TLR7 (0.55) TLR7HDAC1HDAC8HDAC6PIK3CD
SCHEMBL5518286 0.77 TLR7 (0.44) TLR7PIK3CDPIK3CAPIK3CBPIK3CG
SCHEMBL22644581 0.76 TLR7 (0.60) TLR7HDAC1HDAC8HDAC6PIK3CD
SCHEMBL5731967 0.76 TLR7 (0.52) TLR7HDAC1HDAC8HDAC6PIK3CD
SCHEMBL2754047 0.76 TLR7 (0.49) TLR7HDAC1HDAC8HDAC6PIK3CD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8367666-B2 3-carbamoyl-2-pyridone derivatives SHIONOGI & CO., LTD. (JP) 2013-02-05 US disclosed
US-8367666-B2 3-carbamoyl-2-pyridone derivatives SHIONOGI & CO., LTD. (JP) 2013-02-05 US disclosed
US-8178681-B2 methyl 3-methyl-2-{[2-oxo-1-(2-oxo-ethyl)-1,2,5,6,7,8,9,10-octahydro-cycloocta[b]pyridine-3-carbonyl]-amino}-butyrate; cannabinoid receptor agonist; antiinflammatory agent, immunostimulant, analgesic; atopic dermatitis; excellent in photostability, and have excellent transdermal and oral absorbency SHIONOGI & CO., LTD. (JP) 2012-05-15 US disclosed