SCHEMBL5513199

SCHEMBL5513199

O=c1[nH]c(=O)n(F)c2nc[nH]c12

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 7/20 0.58
PDE4A P27815 5/20 0.58
PDE4B Q07343 5/20 0.58
PDE4C Q08493 5/20 0.58
PDE4D Q08499 5/20 0.58
ADORA2B P29275 4/20 0.55
ADORA3 P0DMS8 2/20 0.55
ADORA1 P30542 2/20 0.55
HPGD P15428 1/20 0.55
BLM P54132 1/20 0.55
PDE3A Q14432 1/20 0.55
HSD17B10 Q99714 1/20 0.55
PNP P00491 2/20 0.53
MPO P05164 2/20 0.44
TPO P07202 2/20 0.44
GDA Q9Y2T3 2/20 0.43
ACHE P22303 1/20 0.43
ALDH1A1 P00352 1/20 0.41
ATAD2 Q6PL18 1/20 0.40
PIK3CD O00329 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
3-Methylxanthine SCHEMBL237146 0.78 ADORA2A (0.64) ADORA2APDE4APDE4BPDE4CPDE4D
SCHEMBL18112639 0.78 ADORA2A (0.58) ADORA2APDE4APDE4BPDE4CPDE4D
SCHEMBL864455 0.78 ADORA2A (0.58) ADORA2APDE4APDE4BPDE4CPDE4D
SCHEMBL5515323 0.77 ADORA2A (0.71) ADORA2APDE4APDE4BPDE4CPDE4D
3-Methylxanthine SCHEMBL30753411 0.76 ADORA2A (0.62) ADORA2APDE4APDE4BPDE4CPDE4D
3-Methylxanthine SCHEMBL4020124 0.76 ADORA2A (0.62) ADORA2APDE4APDE4BPDE4CPDE4D
3-Methylxanthine SCHEMBL9317914 0.76 ADORA2A (0.62) ADORA2APDE4APDE4BPDE4CPDE4D
SCHEMBL7466316 0.74 ADORA2A (1.00) ADORA2APDE4APDE4BPDE4CPDE4D
SCHEMBL20653044 0.74 ADORA2A (0.58) ADORA2APDE4APDE4BPDE4CPDE4D
SCHEMBL30171311 0.74 ADORA2A (0.50) ADORA2APDE4APDE4BPDE4CPDE4D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1869011-A2 1H-BENZIMIDAZOLE-4-CARBOXAMIDES SUBSTITUTED WITH A QUATERNARY CARBON AT THE 2-POSITION ARE POTENT PARP INHIBITORS ABBOTT LABORATORIES (US) 2007-12-26 EP claimed
WO-2006110816-A2 1H-BENZIMIDAZOLE-4-CARBOXAMIDES SUBSTITUTED WITH A QUATERNARY CARBON AT THE 2-POSITION ARE POTENT PARP INHIBITORS ABBOTT LABORATORIES (US) 2006-10-19 WO claimed
CN-100478364-C Ethylene polymer and molded article obtained therefrom MITSUI CHEMICALS INC (JP) 2009-04-15 CN disclosed
US-7208559-B2 Ethylened polymer and molded object obtained therefrom MITSUI CHEMICALS, INC. (JP) 2007-04-24 US disclosed
US-20060135712-A1 Ethylened polymer and molded object obtained therefrom MITSUI CHEMICALS, INC. (JP) 2006-06-22 US disclosed
CN-1732189-A Ethylene polymer and molded article obtained therefrom MITSUI CHEMICALS INC (JP) 2006-02-08 CN disclosed