SCHEMBL5513586

SCHEMBL5513586

CNC(=O)c1cc2c(n(Cc3ccc(F)cc3)c1=O)CCCCCC2

nearest known ligand 0.70

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CNR2 P34972 19/20 0.70
CNR1 P21554 18/20 0.70
FAAH O00519 4/20 0.51
ABHD12 Q8N2K0 1/20 0.49
BRD4 O60885 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11922864 0.90 CNR2 (0.71) CNR2CNR1FAAHABHD12
SCHEMBL5508292 0.89 CNR1 (0.67) CNR2CNR1FAAHABHD12
SCHEMBL5513704 0.89 CNR2 (0.56) CNR2CNR1
SCHEMBL5521936 0.87 CNR2 (0.55) CNR2CNR1
SCHEMBL2746302 0.86 CNR2 (0.69) CNR2CNR1FAAH
SCHEMBL5520938 0.85 CNR2 (0.67) CNR2CNR1
SCHEMBL2746521 0.84 CNR1 (0.67) CNR2CNR1FAAHABHD12
SCHEMBL2745483 0.84 CNR1 (0.68) CNR2CNR1FAAH
SCHEMBL5524789 0.84 CNR1 (0.67) CNR2CNR1FAAHABHD12
SCHEMBL2746530 0.83 CNR2 (0.62) CNR2CNR1FAAH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8367666-B2 3-carbamoyl-2-pyridone derivatives SHIONOGI & CO., LTD. (JP) 2013-02-05 US disclosed
US-8178681-B2 methyl 3-methyl-2-{[2-oxo-1-(2-oxo-ethyl)-1,2,5,6,7,8,9,10-octahydro-cycloocta[b]pyridine-3-carbonyl]-amino}-butyrate; cannabinoid receptor agonist; antiinflammatory agent, immunostimulant, analgesic; atopic dermatitis; excellent in photostability, and have excellent transdermal and oral absorbency SHIONOGI & CO., LTD. (JP) 2012-05-15 US disclosed